Danielle Skropeta

Summary

Affiliation: University of Wollongong
Country: Australia

Publications

  1. pmc Kinase inhibitors from marine sponges
    Danielle Skropeta
    School of Chemistry, University of Wollongong, Wollongong, NSW 2522, Australia
    Mar Drugs 9:2131-54. 2011
  2. doi request reprint Deep-sea natural products
    Danielle Skropeta
    School of Chemistry, University of Wollongong, Wollongong, Australia
    Nat Prod Rep 25:1131-66. 2008
  3. doi request reprint The effect of individual N-glycans on enzyme activity
    Danielle Skropeta
    School of Chemistry, University of Wollongong, Wollongong, NSW 2522, Australia
    Bioorg Med Chem 17:2645-53. 2009
  4. doi request reprint N-phenethyl and N-naphthylmethyl isatins and analogues as in vitro cytotoxic agents
    Lidia Matesic
    School of Chemistry, University of Wollongong, Wollongong, NSW 2522, Australia
    Bioorg Med Chem 16:3118-24. 2008
  5. doi request reprint Computational characterisation of the interactions between human ST6Gal I and transition-state analogue inhibitors: insights for inhibitor design
    Andrew Montgomery
    School of Chemistry, Faculty of Science, Medicine and Health, University of Wollongong, Wollongong, NSW, 2522, Australia
    J Mol Recognit 29:210-22. 2016
  6. ncbi request reprint Kinase inhibitory, haemolytic and cytotoxic activity of three deep-water sponges from North Western Australia and their fatty acid composition
    Ana Zivanovic
    School of Chemistry, University of Wollongong, NSW 2500, Australia
    Nat Prod Commun 6:1921-4. 2011
  7. ncbi request reprint c-AMP dependent protein kinase A inhibitory activity of six algal extracts from southeastern Australia and their fatty acid composition
    Ana Zivanovic
    School of Chemistry, University of Wollongong, NSW, 2500, Australia
    Nat Prod Commun 7:923-6. 2012
  8. doi request reprint Parameters affecting the analytical profile of fatty acids in the macroalgal genus Ulva
    Janice I McCauley
    School of Chemistry, Faculty of Science, Medicine, and Health SMAH, University of Wollongong, NSW 2522, Australia Electronic address
    Food Chem 209:332-40. 2016
  9. doi request reprint Advancement of Sialyltransferase Inhibitors: Therapeutic Challenges and Opportunities
    Rémi Szabo
    School of Chemistry, University of Wollongong, Wollongong, NSW, 2522, Australia
    Med Res Rev . 2016
  10. doi request reprint Bioassays for anticancer activities
    Janice McCauley
    School of Chemistry, University of Wollongong, Wollongong, Australia
    Methods Mol Biol 1055:191-205. 2013

Collaborators

Detail Information

Publications11

  1. pmc Kinase inhibitors from marine sponges
    Danielle Skropeta
    School of Chemistry, University of Wollongong, Wollongong, NSW 2522, Australia
    Mar Drugs 9:2131-54. 2011
    ..These compounds, which belong to diverse structural classes, are reviewed herein, and ordered based upon the kinase that they inhibit. Relevant synthetic studies on the marine natural product kinase inhibitors have also been included...
  2. doi request reprint Deep-sea natural products
    Danielle Skropeta
    School of Chemistry, University of Wollongong, Wollongong, Australia
    Nat Prod Rep 25:1131-66. 2008
    ..Relevant synthetic studies on the deep-sea natural products have also been included...
  3. doi request reprint The effect of individual N-glycans on enzyme activity
    Danielle Skropeta
    School of Chemistry, University of Wollongong, Wollongong, NSW 2522, Australia
    Bioorg Med Chem 17:2645-53. 2009
    ....
  4. doi request reprint N-phenethyl and N-naphthylmethyl isatins and analogues as in vitro cytotoxic agents
    Lidia Matesic
    School of Chemistry, University of Wollongong, Wollongong, NSW 2522, Australia
    Bioorg Med Chem 16:3118-24. 2008
    ..The results allowed further development of structure-activity relationships. The compound 5,7-dibromo-N-(1-naphthylmethyl)-1H-indole-2,3-dione 5a was the most potent against U937 cells with an IC(50) value of 0.19 microM...
  5. doi request reprint Computational characterisation of the interactions between human ST6Gal I and transition-state analogue inhibitors: insights for inhibitor design
    Andrew Montgomery
    School of Chemistry, Faculty of Science, Medicine and Health, University of Wollongong, Wollongong, NSW, 2522, Australia
    J Mol Recognit 29:210-22. 2016
    ..Overall, the results obtained from this study provide a rationale for synthetic and biological evaluation of triazole- and carbamate-linked transition-state analogue ST inhibitors as potential new antimetastatic agents...
  6. ncbi request reprint Kinase inhibitory, haemolytic and cytotoxic activity of three deep-water sponges from North Western Australia and their fatty acid composition
    Ana Zivanovic
    School of Chemistry, University of Wollongong, NSW 2500, Australia
    Nat Prod Commun 6:1921-4. 2011
    ....
  7. ncbi request reprint c-AMP dependent protein kinase A inhibitory activity of six algal extracts from southeastern Australia and their fatty acid composition
    Ana Zivanovic
    School of Chemistry, University of Wollongong, NSW, 2500, Australia
    Nat Prod Commun 7:923-6. 2012
    ..Importantly, this study reveals that abundant and readily available marine algae are a new and relatively unexplored source of PKA inhibitory compounds...
  8. doi request reprint Parameters affecting the analytical profile of fatty acids in the macroalgal genus Ulva
    Janice I McCauley
    School of Chemistry, Faculty of Science, Medicine, and Health SMAH, University of Wollongong, NSW 2522, Australia Electronic address
    Food Chem 209:332-40. 2016
    ..High nutrient conditions showed the most desirable FA profile for health, along with the highest total FA content (56mgg(-1) dry weight equivalent) when extracted with an optimised protocol. ..
  9. doi request reprint Advancement of Sialyltransferase Inhibitors: Therapeutic Challenges and Opportunities
    Rémi Szabo
    School of Chemistry, University of Wollongong, Wollongong, NSW, 2522, Australia
    Med Res Rev . 2016
    ....
  10. doi request reprint Bioassays for anticancer activities
    Janice McCauley
    School of Chemistry, University of Wollongong, Wollongong, Australia
    Methods Mol Biol 1055:191-205. 2013
    ..Both assays are highly versatile and can be modified to test against targeted disease processes by using specific kinase enzymes or cell lines. ..
  11. ncbi request reprint N,O-isopropylidenated threonines as tools for peptide cyclization: application to the synthesis of mahafacyclin B
    Nima Sayyadi
    School of Chemistry, The University of Sydney, 2006 NSW, Australia
    Org Lett 7:5497-9. 2005
    ..Incorporation of an N,O-isopropylidenated threonine more than doubles the head-to-tail cyclization yield. The N,O-isopropylidene grouping is then readily disassembled to give the antimalarial cyclic peptide in high yield...