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| neuroprotective agentsSummarySummary: Drugs intended to prevent damage to the brain or spinal cord from ischemia, stroke, convulsions, or trauma. Some must be administered before the event, but others may be effective for some time after. They act by a variety of mechanisms, but often directly or indirectly minimize the damage produced by endogenous excitatory amino acids. Top Publications
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Publications
Blockade of microglial activation is neuroprotective in the 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine mouse model of Parkinson diseaseD C Wu
Department of Neurology, Columbia University, New York, New York 10032, USA
J Neurosci 22:1763-71. 2002..This study demonstrates that microglial-related inflammatory events play a significant role in the MPTP neurotoxic process and suggests that minocycline may be a valuable neuroprotective agent for the treatment of PD...
Role of microglia in inflammation-mediated neurodegenerative diseases: mechanisms and strategies for therapeutic interventionBin Liu
Neuropharmacology Section, Laboratory of Pharmacology and Chemistry, National Institute of Environmental Health Sciences, National Institutes of Health, Research Triangle Park, North Carolina 27709, USA
J Pharmacol Exp Ther 304:1-7. 2003..In addition, we also discuss novel approaches to potential therapeutic strategies...
ERK activation by the polyphenols fisetin and resveratrol provides neuroprotection in multiple models of Huntington's diseasePamela Maher
Department of Cellular Neurobiology, The Salk Institute for Biological Studies, La Jolla, CA 92037, USA
Hum Mol Genet 20:261-70. 2011..Thus, fisetin, resveratrol and related compounds might be useful for the treatment of HD by virtue of their unique ability to activate ERK...
Neuroprotection for ischemic stroke: past, present and futureMyron D Ginsberg
Department of Neurology D4 5, University of Miami Miller School of Medicine, Miami, FL 33101, USA
Neuropharmacology 55:363-89. 2008..This review presents a close survey of the most extensively evaluated neuroprotective agents and classes and considers both the strengths and weakness of the pre-clinical evidence as well as the ..
Minocycline, a tetracycline derivative, is neuroprotective against excitotoxicity by inhibiting activation and proliferation of microgliaT Tikka
A. I. Virtanen Institute for Molecular Sciences, University of Kuopio, FIN-70211 Kuopio, Finland
J Neurosci 21:2580-8. 2001..These findings indicate that the proliferation and activation of microglia contributes to excitotoxicity, which is inhibited by minocycline, an antibiotic used in severe human infections...
Randomized, double-blind trial of glial cell line-derived neurotrophic factor (GDNF) in PDJ G Nutt
Oregon Health and Science University, Portland 97201 3098, USA
Neurology 60:69-73. 2003..To assess the safety, tolerability, and biological activity of glial cell line-derived neurotrophic factor (GDNF) administered by an implanted intracerebroventricular (ICV) catheter and access port in advanced PD...
Use of anti-aging herbal medicine, Lycium barbarum, against aging-associated diseases. What do we know so far?Raymond Chuen Chung Chang
Laboratory of Neurodegenerative Diseases, Department of Anatomy, LKS Faculty of Medicine, The University of Hong Kong, Pokfulam, Hong Kong SAR, China
Cell Mol Neurobiol 28:643-52. 2008..barbarum. We hope that new findings for L. barbarum will pave a new avenue for the use of Chinese medicine in modern evidence-based medicine...
1,026 experimental treatments in acute strokeMalcolm R Macleod
Neuroscience Lab, Department of Medicine, University of Melbourne, Austin Health, Heidelberg, VIC 3084, Australia
Ann Neurol 59:467-77. 2006..This may partially explain the slow progress in developing treatments. Greater rigor in the conduct, reporting, and analysis of animal data will improve the transition of scientific advances from bench to bedside...
Hydrogen sulfide protects neurons from oxidative stressYuka Kimura
National Institute of Neuroscience, Kodaira, Tokyo, Japan
FASEB J 18:1165-7. 2004..Cystine (cysteine) is the rate-limiting substrate of glutathione synthesis. These observations reveal that H2S protects neurons from oxytosis by increasing the production of the antioxidant glutathione...
Beta-lactam antibiotics offer neuroprotection by increasing glutamate transporter expressionJeffrey D Rothstein
Department of Neurology, Johns Hopkins University, Baltimore, Maryland 21287, USA
Nature 433:73-7. 2005..Thus these studies provide a class of potential neurotherapeutics that act to modulate the expression of glutamate neurotransmitter transporters via gene activation...
Involvement of ROS in BBB dysfunctionPamela B L Pun
Defence Medical and Environmental Research Institute, DSO National Laboratories, Singapore
Free Radic Res 43:348-64. 2009..This review explores some of the pathways both upstream and downstream of ROS that have been implicated in increased BBB permeability and discusses the role of ROS and antioxidants in neuropathology...
Minocycline prevents nigrostriatal dopaminergic neurodegeneration in the MPTP model of Parkinson's diseaseY Du
Departmens of Pharmacology and Toxicology, Indiana University School of Medicine, Indianapolis, IN 46202, USA
Proc Natl Acad Sci U S A 98:14669-74. 2001..Thus, NO appears to play an important role in MPTP neurotoxicity. Neuroprotective tetracyclines may be effective in preventing or slowing the progression of Parkinson's and other neurodegenerative diseases...
Erythropoietin crosses the blood-brain barrier to protect against experimental brain injuryM L Brines
The Kenneth S Warren Laboratories, 765 Old Saw Mill River Road, Tarrytown, NY 10591, USA
Proc Natl Acad Sci U S A 97:10526-31. 2000..Given r-Hu-EPO's excellent safety profile, clinical trials evaluating systemically administered r-Hu-EPO as a general neuroprotective treatment are warranted...
Tripchlorolide protects neuronal cells from microglia-mediated beta-amyloid neurotoxicity through inhibiting NF-kappaB and JNK signalingXiao Dong Pan
Department of Neurology, Union Hospital of Fujian Medical University, Fuzhou, Fujian, People s Republic of China
Glia 57:1227-38. 2009..Therefore, T4 may be an effective agent in modulating neuroinflammatory process in AD...
ProTECT: a randomized clinical trial of progesterone for acute traumatic brain injuryDavid W Wright
Department of Emergency Medicine, School of Medicine of Emory University, Atlanta, GA, USA
Ann Emerg Med 49:391-402, 402.e1-2. 2007..Laboratory evidence indicates that progesterone has potent neuroprotective effects. We conducted a pilot clinical trial to assess the safety and potential benefit of administering progesterone to patients with acute traumatic brain injury...
Neuroprotective effects of Lycium barbarum Lynn on protecting retinal ganglion cells in an ocular hypertension model of glaucomaHiu Chi Chan
Department of Anatomy, Faculty of Medicine, The University of Hong Kong, Pokfulam, Hong Kong SAR
Exp Neurol 203:269-73. 2007..barbarum against neurodegeneration in the retina of rat OH model. The results demonstrate that this extract may be a potential candidate for the development of neuroprotective drug against the loss of RGCs in glaucoma...
The neuroprotective effect of xenon administration during transient middle cerebral artery occlusion in miceH Mayumi Homi
Department of Anesthesiology (Multidisciplinary Neuroprotection Laboratories, Duke University Medical Center, Durham, North Carolina, USA
Anesthesiology 99:876-81. 2003..0009). CONCLUSIONS: In this model of transient focal cerebral ischemia, xenon administration improved both functional and histologic outcome...
Minocycline delays disease onset and mortality in a transgenic model of ALSLudo Van Den Bosch
Laboratory for Neurobiology, Campus Gasthuisberg, Herestraat 49, B-3000 Leuven, Belgium
Neuroreport 13:1067-70. 2002..These results demonstrate that interference with immuno-inflammatory responses has a beneficial effect in the ALS mice model, suggesting this to be a potential new strategy to treat ALS...
Green tea epigallocatechin-3-gallate (EGCG) reduces beta-amyloid mediated cognitive impairment and modulates tau pathology in Alzheimer transgenic miceKavon Rezai-Zadeh
Rashid Laboratory for Developmental Neurobiology, Silver Child Development Center, Department of Psychiatry and Behavioral Medicine, and Department of Neurosurgery, University of South Florida, Tampa, FL 33613, USA
Brain Res 1214:177-87. 2008..Taken together, these data further the notion of EGCG dietary supplementation as a potentially safe and effective prophylaxis for Alzheimer's disease...
Edaravone prevents kainic acid-induced neuronal deathRyohei Miyamoto
Department of Pediatrics, Osaka Medical College, Japan
Brain Res 1209:85-91. 2008..Patients who develop status epilepticus are unlikely to receive adequate antioxidant therapy before the onset, so it is an advantage that Ed can prevent neuronal death even when administered after seizures...
Role for matrix metalloproteinase 9 after focal cerebral ischemia: effects of gene knockout and enzyme inhibition with BB-94M Asahi
Department of Neurology, Massachusetts General Hospital, and Harvard Medical School, Charlestown 02129, USA
J Cereb Blood Flow Metab 20:1681-9. 2000..These data demonstrate that MMP-9 plays a deleterious role in the development of brain injury after focal ischemia...
Minocycline treatment in acute stroke: an open-label, evaluator-blinded studyY Lampl
Department of Neurology, Edith Wolfson Medical Center, Holon 58100, Israel
Neurology 69:1404-10. 2007..Ischemic animal model studies have shown a neuroprotective effect of minocycline...
Neuronal estrogen receptor-alpha mediates neuroprotection by 17beta-estradiolJoachim G Elzer
Division of Molecular Biology of the Cell 1, German Cancer Research Center, Heidelberg, Germany
J Cereb Blood Flow Metab 30:935-42. 2010..We conclude that neuronal ER alpha in female and male mice mediates neuroprotective estrogen effects in an in vivo mouse model of stroke, whereas microglial ER alpha is dispensable...
Neuroprotection in the newborn infantFernando F Gonzalez
Department of Pediatrics, University of California, 521 Parnassus Avenue, C215, Box 0663, San Francisco, CA 94143, USA
Clin Perinatol 36:859-80, vii. 2009..More recent evidence suggests combined therapy may optimize repair, decreasing cell injury while increasing newly born cells...
Neuroprotection by baicalein in ischemic brain injury involves PTEN/AKT pathwayChao Liu
Department of Pharmacology, Pharmaceutical College, Xianning University, Xianning, China
J Neurochem 112:1500-12. 2010..Together, these findings provide evidence that Bai protects neurons against ischemia injury and this neuroprotective effect involves PI3K/Akt and PTEN pathway...
Targeting the p53 pathway to protect the neonatal ischemic brainCora H Nijboer
Laboratory of Neuroimmunology and Developmental Origins of Disease, University Medical Center Utrecht, Utrecht, The Netherlands
Ann Neurol 70:255-64. 2011..To investigate whether inhibition of mitochondrial p53 association using pifithrin-μ (PFT-μ) represents a potential novel neuroprotective strategy to combat perinatal hypoxic-ischemic (HI) brain damage...
Neuropharmacological and pharmacokinetic properties of berberine: a review of recent researchMinzhong Ye
Department of Pharmacology and Toxicology, School of Pharmaceutical Sciences, Sun Yat Sen University, Guangzhou, PR China
J Pharm Pharmacol 61:831-7. 2009..This review summarizes recent research on the neuropharmacological and pharmacokinetic properties of berberine, an isoquinoline alkaloid extracted from Coptidis rhizoma...
Neuroprotectin D1 (NPD1): a DHA-derived mediator that protects brain and retina against cell injury-induced oxidative stressNicolas G Bazan
LSU Neuroscience Center and Department of Opthamology, Louisiana State University Health Sciences Center School of Medicine, New Orleans 70112, USA
Brain Pathol 15:159-66. 2005....
Erythropoietin improves histological and functional outcomes after traumatic brain injury in mice in the absence of the neural erythropoietin receptorYe Xiong
Department of Neurosurgery, Henry Ford Health System, Detroit, Michigan 48202, USA
J Neurotrauma 27:205-15. 2010..These data demonstrate that EPO significantly provides neuroprotection following TBI, even in the absence of EPOR in the neural cells, suggesting that its therapeutic benefits may be mediated through vascular protection...
Reproductive age modulates the impact of focal ischemia on the forebrain as well as the effects of estrogen treatment in female ratsAmutha Selvamani
Department of Neuroscience and Experimental Therapeutics, Texas A and M Health Science Center, College Station, TX 77843 1114, USA
Neurobiol Aging 31:1618-28. 2010....
Nuclear factor E2-related factor 2-dependent antioxidant response element activation by tert-butylhydroquinone and sulforaphane occurring preferentially in astrocytes conditions neurons against oxidative insultAndrew D Kraft
School of Pharmacy, University of Wisconsin, Madison, Wisconsin 53705 2222, USA
J Neurosci 24:1101-12. 2004..Strikingly, the change in neuronal gene expression after tBHQ treatment was dependent on Nrf2 activity in the astrocytes. This suggests that Nrf2-dependent genetic changes alter neuron-glia interactions resulting in neuroprotection...
Neurotrophin roles in retinal ganglion cell survival: lessons from rat glaucoma modelsElaine C Johnson
The Kenneth C Swan Ocular Neurobiology Laboratory, Casey Eye Institute, Ceres, Oregon Health and Science University, Portland, OR 97239, USA
Exp Eye Res 88:808-15. 2009..The examination of these studies in this review reveals a number of consistent observations and provides direction for further investigations of this hypothesis...
Sex differences in minocycline-induced neuroprotection after experimental strokeJun Li
Department of Neurology, University of Connecticut Health Center, Farmington, Connecticut 06030, USA
J Cereb Blood Flow Metab 29:670-4. 2009..Clinical trials must consider possible sex differences in the response to neuroprotective agents, if we hope to translate promising therapies to stroke patients of both sexes.
Neuronal PPARgamma deficiency increases susceptibility to brain damage after cerebral ischemiaXiurong Zhao
Stroke Program, Department of Neurology, University of Texas, Houston, Medical School, Houston, Texas 77030, USA
J Neurosci 29:6186-95. 2009..Therefore, we conclude that PPARgamma in neurons play an essential protective function and that PPARgamma agonists may have utility in neuronal self-defense, in addition to their well established anti-inflammatory effect...
Neuroprotective effects of curcuminGreg M Cole
Greater Los Angeles Veterans Affairs Healthcare System, Geriatric Research, Education, and Clinic Center, Sepulveda, CA 91343, USA
Adv Exp Med Biol 595:197-212. 2007..Promising results have already led to ongoing pilot clinical trials...
Modulation of the endocannabinoid system: neuroprotection or neurotoxicity?Christopher J Fowler
Department of Pharmacology and Clinical Neuroscience, Umea University, SE 901 87 Umea, Sweden
Exp Neurol 224:37-47. 2010....
Neuroprotective effects of creatine in a transgenic animal model of amyotrophic lateral sclerosisP Klivenyi
Neurochemistry Laboratory, Neurology Service, Massachusetts General Hospital and Harvard Medical School, Boston 02118, USA
Nat Med 5:347-50. 1999..Creatine administration protected G93A transgenic mice from increases in biochemical indices of oxidative damage. Therefore, creatine administration may be a new therapeutic strategy for ALS...
Nutraceutical antioxidants as novel neuroprotective agentsNatalie A Kelsey
Department of Biological Sciences and Eleanor Roosevelt Institute, University of Denver, Denver, Colorado 80208, USA
Molecules 15:7792-814. 2010..Here, we review the literature pertaining to these various classes of nutraceutical antioxidants and discuss their potential therapeutic value in neurodegenerative diseases...
Neuroprotective strategies involving ROS in Alzheimer diseaseMagali Dumont
Department of Neurology and Neuroscience, Weill Cornell Medical College, New York, NY 10065, USA
Free Radic Biol Med 51:1014-26. 2011..Nonetheless, there is still hope for improved compounds that would better target pathways implicated in ROS production. In fact, facilitating the endogenous antioxidant system by modulating transcription has great promise for AD therapy...
Monoamine oxidase inhibitors as neuroprotective agents in age-dependent neurodegenerative disordersMakoto Naoi
Department of Neurosciences, Gifu International Institute of Biotechnology, 1 1 Nakafudogaoka, Kakamigahara, Gifu 504 0838, Japan
Curr Pharm Des 16:2799-817. 2010..the inhibitors of type B monoamine oxidase, such as selegiline and rasagiline, are the most promising neuroprotective agents to date. These inhibitors protect neuronal cells against cell death induced in cellular and animal models...
Alzheimer's disease: the pros and cons of pharmaceutical, nutritional, botanical, and stimulatory therapies, with a discussion of treatment strategies from the perspective of patients and practitionersKeith A Wollen
Psychology Department of Washington State University, USA
Altern Med Rev 15:223-44. 2010..Approaches that target several dysfunctions simultaneously and that emphasize nutritional, botanical, and stimulatory therapies may offer the most benefit at this time...
Tetrahydrocurcumin confers protection against amyloid β-induced toxicityShilpa Mishra
National Brain Research Centre, Manesar, Haryana, India
Neuroreport 22:23-7. 2011..Thus, THC confers protection against amyloid-β-induced toxicity, and the antioxidant activity may contribute to its protective effect...
Neuroprotective effect of Bax-inhibiting peptide on neonatal brain injuryXiaoyang Wang
Department of Physiology, Perinatal Center, Sahlgrenska Academy, University of Gothenburg, Box 432, S 405 30 Gothenburg, Sweden
Stroke 41:2050-5. 2010..The aim of this study was to evaluate the neuroprotective effect of a cell-penetrating Bax-inhibiting peptide (BIP) on neonatal mouse HI brain injury...
Peroxisome proliferator-activated receptor gamma agonists as neuroprotective agentsRavinder K Kaundal
Department of Pharmacology and Toxicology of the National Institute of Pharmaceutical Education and Research NIPER, Mohali, Punjab, India
Drug News Perspect 23:241-56. 2010..This article discusses evidence and mechanisms supporting the neuroprotective effects of PPARgamma agonists in central nervous system disorders...
Lycium barbarum polysaccharides reduce neuronal damage, blood-retinal barrier disruption and oxidative stress in retinal ischemia/reperfusion injurySuk Yee Li
Eye Institute, Li Ka Shing Faculty of Medicine, The University of Hong Kong, Hong Kong
PLoS ONE 6:e16380. 2011..The present study suggests that LBP may have a neuroprotective role to play in ocular diseases for which I/R is a feature...
Neuroprotective effects of female gonadal steroids in reproductively senescent female ratsN J Alkayed
Department of Anesthesiology, Division of Comparative Medicine, Johns Hopkins University School of Medicine, Baltimore, MD, USA
Stroke 31:161-8. 2000....
Heme oxygenase 1, beneficial role in permanent ischemic stroke and in Gingko biloba (EGb 761) neuroprotectionZ A Shah
Department of Medicinal and Biological Chemistry, College of Pharmacy and Pharmaceutical Sciences, University of Toledo, Toledo, OH 43614, USA
Neuroscience 180:248-55. 2011..Together, these results suggest that HO1 plays, at least in part, an important role in the neuroprotective mechanism of EGb 761 and in delayed ischemia. Targeting this pathway could lead to neuroprotective agents against ischemic stroke.
Inhibition of extracellular signal-regulated kinases 1/2 provides neuroprotection in spinal cord ischemia/reperfusion injury in rats: relationship with the nuclear factor-kappaB-regulated anti-apoptotic mechanismsKang Lu
Department of Neurosurgery, E Da Hospital, I Shou University, Kaohsiung 824, Taiwan
J Neurochem 114:237-46. 2010..Future research should focus on the possible cross-talk between the MEK/ERK pathway and the NF-kappaB transcriptional cascade...
Actions of estrogens on glial cells: Implications for neuroprotectionMaria Angeles Arevalo
Instituto Cajal, CSIC, Madrid, Spain
Biochim Biophys Acta 1800:1106-12. 2010..Therefore, glial cells are important players in the neuroprotective and reparative mechanisms of estrogenic compounds...
Fish consumption, long-chain omega-3 fatty acids and risk of cognitive decline or Alzheimer disease: a complex associationMajid Fotuhi
Center for Memory and Brain Health, LifeBridge Health Brain and Spine Institute, Sinai Hospital of Baltimore, Baltimore, MD 21209, USA
Nat Clin Pract Neurol 5:140-52. 2009..Large clinical trials of extended duration should help to provide definitive answers...
Neuroprotection by BDNF against glutamate-induced apoptotic cell death is mediated by ERK and PI3-kinase pathwaysR D Almeida
Center for Neuroscience and Cell Biology and Department of Zoology, University of Coimbra, 3004-517 Coimbra, Portugal
Cell Death Differ 12:1329-43. 2005..The results indicate that the protective effect of BDNF in hippocampal neurons against glutamate toxicity is mediated by the PI3-K and the Ras/MAPK signaling pathways, and involves a long-term change in protein synthesis...
Nerve growth factor survival signaling in cultured hippocampal neurons is mediated through TrkA and requires the common neurotrophin receptor P75C Culmsee
Institut fur Pharmakologie und Toxikologie, Philipps Universitat Marburg, Ketzerbach 63, 35032, Marburg, Germany
Neuroscience 115:1089-108. 2002..Overall, our results indicate an essential role for p75NTR in supporting NGF-triggered TrkA signaling pathways mediating neuronal survival in hippocampal neurons...
The therapeutic window after spinal cord injury can accommodate T cell-based vaccination and methylprednisolone in ratsAntonio Ibarra
Department of Neurobiology, The Weizmann Institute of Science, 76100 Rehovot, Israel
Eur J Neurosci 19:2984-90. 2004..These results demonstrate that the therapeutic window after SCI can accommodate immediate administration of MP plus a delayed therapeutic vaccination...
Preclinical development of neurosteroids as neuroprotective agents for the treatment of neurodegenerative diseasesP A Lapchak
Department of Neuroscience, University of California-San Diego, La Jolla, California 92093-0624, USA
Int Rev Neurobiol 46:379-97. 2001..2000), their potential therapeutic benefits may be extended to include the treatment of other neurodegenerative diseases not directly linked to excitotoxicity...
Post-ischemic helium provides neuroprotection in rats subjected to middle cerebral artery occlusion-induced ischemia by producing hypothermiaHelene N David
NNOXe Pharmaceuticals, Quebec City, Quebec, Canada
J Cereb Blood Flow Metab 29:1159-65. 2009..In this study, we show that helium at 75 vol% produces neuroprotection and improvement of neurologic outcome in rats subjected to transient MCAO by producing hypothermia on account of its high specific heat as compared with air...
The potential value of natural antioxidative treatment in glaucomaM Mozaffarieh
Department of Ophthalmology, University Hospital Basel, Switzerland
Surv Ophthalmol 53:479-505. 2008..Anthocyanosides (bilberries) owe their antioxidant effects to their particular chemical structure. Other antioxidants include ubiquinone and melatonin...
Argon: neuroprotection in in vitro models of cerebral ischemia and traumatic brain injuryPhilip D Loetscher
Department of Anesthesiology, University Hospital of the RWTH Aachen, Aachen, Germany
Crit Care 13:R206. 2009..Since traumatic brain injury and stroke are widespread and generate an enormous economic and social burden, we investigated the possible neuroprotective effect in in vitro models of traumatic brain injury and cerebral ischemia...
The flavonoid baicalin counteracts ischemic and oxidative insults to retinal cells and lipid peroxidation to brain membranesS H Jung
Nuffield Laboratory of Ophthalmology, Oxford University, John Radcliffe Hospital, Oxford OX3 9DU, UK
Neurochem Int 53:325-37. 2008..Significantly, the negative insult of serum withdrawal on RGC-5 cell survival was blunted by baicalin but not by EGCG revealing the different properties of the two flavonoids...
Role of creatine and phosphocreatine in neuronal protection from anoxic and ischemic damageM Balestrino
Department of Neurological and Vision Sciences, University of Genova, Italy
Amino Acids 23:221-9. 2002..Accordingly, preliminary data show that creatine pretreatment decreases ischemic damage in vivo...
Pharmacological neuroprotection for glaucomaGlyn Chidlow
Ophthalmic Research Laboratories, South Australian Institute of Ophthalmology, Hanson Institute, Adelaide, South Australia, Australia
Drugs 67:725-59. 2007....
Hydrogen sulfide is a mediator of cerebral ischemic damageKun Qu
Department of Pharmacology, Yong Loo Lin School of Medicine, National University of Singapore, Kent Ridge, Singapore
Stroke 37:889-93. 2006..CONCLUSIONS: The present results strongly suggest that H2S plays a part in cerebral ischemic damage after stroke. Inhibition of H2S synthesis should be investigated for its potential as a novel neuroprotective stroke therapy...
Cystine/glutamate exchange modulates glutathione supply for neuroprotection from oxidative stress and cell proliferationAndy Y Shih
Kinsmen Laboratory of Neurological Research and Brain Research Center, University of British Columbia, Vancouver, British Columbia, Canada V6T 1Z3
J Neurosci 26:10514-23. 2006..Furthermore, xCT is critical for cell proliferation during development in vitro and possibly in vivo...
Neuroprotection in transient focal brain ischemia after delayed intravenous administration of brain-derived neurotrophic factor conjugated to a blood-brain barrier drug targeting systemY Zhang
Department of Medicine, University of California at Los Angeles School of Medicine, Los Angeles, CA 90095-1682, USA
Stroke 32:1378-84. 2001..The neuroprotection is long lasting and persists for at least 7 days after a 1-hour middle cerebral artery occlusion...
Multifunctional activities of green tea catechins in neuroprotection. Modulation of cell survival genes, iron-dependent oxidative stress and PKC signaling pathwaySilvia A Mandel
Eve Topf and USA National Parkinson Foundation Centers of Excellence for Neurodegenerative Diseases Research, Technion-Faculty of Medicine, Haifa, Israel
Neurosignals 14:46-60. 2005..In particular, their transitional metal (iron and copper) chelating property and inhibition of oxidative stress...
Neuroprotective strategies for basal ganglia degeneration: Parkinson's and Huntington's diseasesT Alexi
Research Centre for Developmental Medicine and Biology, School of Medicine, University of Auckland, New Zealand
Prog Neurobiol 60:409-70. 2000..Considerable research has been done on testing a large array of neuroprotective agents using animal models which mimic these disorders...
Peptide-mediated protection from ethanol-induced neural tube defectsShao Yu Chen
Bowles Center for Alcohol Studies and Department of Cell and Developmental Biology, University of North Carolina, Chapel Hill, NC 27599 7178, USA
Dev Neurosci 27:13-9. 2005..These findings demonstrate the ability of NAP and SAL to prevent ethanol-induced NTDs and support the hypothesis that ethanol teratogenesis is caused in part by ethanol inhibition of L1-mediated cell adhesion...
Atorvastatin reduces neurological deficit and increases synaptogenesis, angiogenesis, and neuronal survival in rats subjected to traumatic brain injuryDunyue Lu
Department of Neurosurgery, Henry Ford Health Sciences Center, Detroit, MI 48202, USA
J Neurotrauma 21:21-32. 2004..The results suggest that atorvastatin may provide beneficial effects in experimental TBI...
Neuroprotective effects of grape seed extract on neuronal injury by inhibiting DNA damage in the gerbil hippocampus after transient forebrain ischemiaIn Koo Hwang
Department of Anatomy, College of Medicine, Hallym University, Chunchon, 200-702, South Korea
Life Sci 75:1989-2001. 2004..Therefore, these results suggest that GSE can protect ischemic neuronal damage by inhibiting DNA damage after transient forebrain ischemia...
EGCG remodels mature alpha-synuclein and amyloid-beta fibrils and reduces cellular toxicityJan Bieschke
Max Delbrueck Center for Molecular Medicine, Robert Roessle Strasse 10, 13125 Berlin Buch, Germany
Proc Natl Acad Sci U S A 107:7710-5. 2010..These findings suggest that EGCG is a potent remodeling agent of mature amyloid fibrils...
Dose dependence and therapeutic window for the neuroprotective effects of curcumin in thromboembolic model of ratPreeti Dohare
Division of Pharmacology, Central Drug Research Institute, Lucknow 226001, India
Behav Brain Res 193:289-97. 2008....
Valproic acid-mediated neuroprotection and regeneration in injured retinal ganglion cellsJulia Biermann
University Eye Hospital Freiburg, Freiburg im Breisgau, Germany
Invest Ophthalmol Vis Sci 51:526-34. 2010..The authors investigated whether VPA delays retinal ganglion cell (RGC) death and enhances axonal regeneration after optic nerve crush (ONC). Furthermore, potential molecular targets involved in VPA-mediated protection were analyzed...
Protective effects of estrogen and selective estrogen receptor modulators in the brainKrishnan M Dhandapani
Institute of Molecular Medicine and Genetics, Program in Neurobiology, and Department of Neurology, Medical College of Georgia, Augusta, Georgia 30912, USA
Biol Reprod 67:1379-85. 2002..The role of other potential mediatory factors such as growth factors and the possibility of an astrocyte role in neuroprotection is also discussed...
Neuroprotective effects of resveratrol against traumatic brain injury in immature ratsUlker Sonmez
Department of Histology and Embryology, School of Medicine, Dokuz Eylul University Inciralti, TR 35340 Izmir, Turkey
Neurosci Lett 420:133-7. 2007..These results show that acute treatment of resveratrol has a neuroprotective role against trauma induced hippocampal neuron loss and associated cognitive impairment in rats...
Prevention of MPTP (N-methyl-4-phenyl-1,2,3,6-tetrahydropyridine) dopaminergic neurotoxicity in mice by chronic lithium: involvements of Bcl-2 and BaxMoussa B H Youdim
Eve Topf and National Parkinson Foundation Centers of Excellence for Neurodegenerative Diseases Research, Faculty of Medicine, Technion, Efron Street, P O Box 9697, Haifa 31096, Israel
Neuropharmacology 46:1130-40. 2004..The neuroprotective action of lithium in this model of Parkinson's disease has been attributed to its antiapoptotic activity which among other factors includes induction of Bcl-2 and reduction of Bax...
Docosahexaenoic acid provides protection from impairment of learning ability in Alzheimer's disease model ratsMichio Hashimoto
Department of Physiology, Shimane Medical University, Izumo, Japan
J Neurochem 81:1084-91. 2002..Docosahexaenoic acid is thus a possible prophylactic means for preventing the learning deficiencies of Alzheimer's disease...
Neuroprotective properties of statins in cerebral ischemia and strokeC J Vaughan
Division of Cardiology, Department of Medicine, Weill Medical College of Cornell University, The New York Presbyterian Hospital, New York, NY 10021, USA
Stroke 30:1969-73. 1999..In this article, we review the emerging evidence that statins have beneficial effects within the cerebral circulation and brain parenchyma during ischemic stroke and reperfusion...
The neuroprotective properties of calorie restriction, the ketogenic diet, and ketone bodiesMarwan Maalouf
Department of Neurobiology, David Geffen School of Medicine, University of California, 63 323 CH5, Box 951763, Los Angeles, CA 90095 1763, USA
Brain Res Rev 59:293-315. 2009..The present review summarizes the neuroprotective effects of calorie restriction, of the ketogenic diet and of ketone bodies, and compares their putative mechanisms of action...
Neuroprotective actions of brain aromataseColin J Saldanha
Department of Biological Sciences, Lehigh University, Bethlehem, PA 18015, United States
Front Neuroendocrinol 30:106-18. 2009....
CEP-1347 reduces mutant huntingtin-associated neurotoxicity and restores BDNF levels in R6/2 miceBarbara L Apostol
Department of Psychiatry and Human Behavior, University of California, Irvine, CA 92697, USA
Mol Cell Neurosci 39:8-20. 2008..These studies suggest a novel therapeutic approach for a currently untreatable neurodegenerative disease, HD, via CEP-1347 up-regulation of BDNF...
The hematopoietic factor granulocyte-colony stimulating factor improves outcome in experimental spinal cord injuryClaudia Pitzer
Sygnis Bioscience, Im Neuenheimer Feld, Heidelberg, Germany
J Neurochem 113:930-42. 2010..We show that G-CSF improves outcome after experimental SCI by counteracting apoptosis, and enhancing connectivity in the injured spinal cord. We conclude that G-CSF constitutes a promising and feasible new therapy option for SCI...
Cyanine dyes attenuate cerebral ischemia and reperfusion injury in ratsSatomi Koya-Miyata
Biomedical Institute, Research Center, Hayashibara Biochemical Laboratories, Inc
Biol Pharm Bull 33:1872-7. 2010..These results suggest that NK-4 and NK-150 effectively prevented ischemia-induced brain injury through their potent neurotrophin-like activity as well as antioxidative activity...
Current and future disease-modifying therapies in multiple sclerosisS Y Lim
University of Nottingham, UK
Int J Clin Pract 64:637-50. 2010..It is also worth noting the evidence for starting DMT in patients with clinically isolated syndrome, whereby early treatment has shown to delay the onset of clinically definite MS in separate phase III studies...
Quercetin activates AMP-activated protein kinase by reducing PP2C expression protecting old mouse brain against high cholesterol-induced neurotoxicityJun Lu
Key Laboratory for Biotechnology on Medicinal Plants of Jiangsu Province, School of Life Science, Xuzhou Normal University, Xuzhou 221116, Jiangsu Province, P R China
J Pathol 222:199-212. 2010..These results suggest that AMPK activated by quercetin may be a potential target to enhance the resistance of neurons to age-related diseases...
Prion protein attenuates excitotoxicity by inhibiting NMDA receptorsHouman Khosravani
Department of Physiology and Biophysics, Hotchkiss Brain Institute, University of Calgary, Calgary T2N4N1, Canada
J Cell Biol 181:551-65. 2008..Thus, native PrP(C) mediates an important neuroprotective role by virtue of its ability to inhibit NR2D subunits...
Heat shock protein 90 mediates cytoprotection by H₂S against chemical hypoxia-induced injury in PC12 cellsJin Lan Meng
Department of Physiology, Zhongshan Medical College, China
Clin Exp Pharmacol Physiol 38:42-9. 2011..01) and increasing ROS production. 7. The findings of the present study provide novel evidence that Hsp90 mediates H₂S-induced neuroprotection against chemical hypoxia-induced injury via anti-oxidant and anti-apoptotic effects...
Protection of mouse photoreceptors by survival factors in retinal degenerationsM M LaVail
Department of Anatomy, University of California, San Francisco 94143 0730, USA
Invest Ophthalmol Vis Sci 39:592-602. 1998....
Alpha2 adrenergic modulation of NMDA receptor function as a major mechanism of RGC protection in experimental glaucoma and retinal excitotoxicityCun Jian Dong
Department of Biological Sciences, Allergan Pharmaceuticals, Irvine, California 92612, USA
Invest Ophthalmol Vis Sci 49:4515-22. 2008..In this study, the authors investigated the neural mechanism that may underlie alpha2 neuroprotection of RGCs...
Neuroprotective activities of CD4+CD25+ regulatory T cells in an animal model of Parkinson's diseaseAshley D Reynolds
Center for Neurovirology and Neurodegenerative Disorders, Department of Pharmacology and Experimental Neuroscience, University of Nebraska Medical Center, Omaha, NE 68198 5880, USA
J Leukoc Biol 82:1083-94. 2007..This neuroprotection was achieved through modulation of microglial oxidative stress and inflammation. As Tregs can be modulated in vivo, these data strongly support the use of such immunomodulatory strategies to treat PD...
TNF-alpha-mediates neuroprotection against glutamate-induced excitotoxicity via NF-kappaB-dependent up-regulation of K2.2 channelsAmalia M Dolga
Department of Molecular Neurobiology, University of Groningen, Haren, The Netherlands
J Neurochem 107:1158-67. 2008..We conclude that treatment of primary cortical neurons with TNF-alpha leads to increased K(Ca)2.2 channel expression which renders neurons more resistant to excitotoxic cell death...
Anticonvulsant and neuroprotective effects of the novel calcium antagonist NP04634 on kainic acid-induced seizures in ratsJose A Morales-Garcia
Instituto de Investigaciones Biomedicas, Consejo Superior de Investigaciones Cientificas Universidad Autonoma de Madrid, and Centro de Investigación Biomédica en Red sobre Enfermedades neurodegenerativas, Madrid, Spain
J Neurosci Res 87:3687-96. 2009..Also, NP04634 prevented the loss of hippocampal CA1 and CA3 pyramidal neurons and reduced the gliosis induced by KA. These results point to a potential anticonvulsant and neuroprotective role for NP04634...
Sample size estimates for clinical trials of vasospasm in subarachnoid hemorrhageKurt T Kreiter
Biogen Idec, Wellesley, MA, USA
Stroke 40:2362-7. 2009....
Inhibitory effect of fucoidan on nitric oxide production in lipopolysaccharide-activated primary microgliaYan qiu Cui
Key Laboratory of Neurodegenerative Diseases of Ministry of Education, Capital Medical University, Beijing, China
Clin Exp Pharmacol Physiol 37:422-8. 2010..The results also suggest that this inhibitory action of fucoidan involves suppression of p38 and ERK phosphorylation...
A nanomedicine transports a peptide caspase-3 inhibitor across the blood-brain barrier and provides neuroprotectionHulya Karatas
Department of Neurology, Faculty of Medicine and Institute of Neurological Sciences and Psychiatry, Hacettepe University, Ankara, Turkey
J Neurosci 29:13761-9. 2009..Thus, chitosan nanospheres open new and exciting opportunities for brain delivery of biologically active peptides that are useful for the treatment of CNS disorders...
Magnesium sulphate in the management of patients with aneurysmal subarachnoid haemorrhage: a meta-analysis of prospective controlled trialsLi Ma
Department of Neurosurgery, Second Affiliated Hospital, College of Medicine, Zhejiang University, PR China
Brain Inj 24:730-5. 2010..A meta-analysis was conducted to assess the effectiveness and safety of intravenous magnesium therapy in patients with aneurysmal subarachnoid haemorrhage (SAH). Research design: Meta-analysis...
Tamoxifen mediated estrogen receptor activation protects against early impairment of hippocampal neuron excitability in an oxygen/glucose deprivation brain slice ischemia modelHuaqiu Zhang
Department of Neurosurgery, Tongji Hospital, Tongji Medical College, Huazhong, University of Science and Technology, Wuhan, 430030, PR China
Brain Res 1247:196-211. 2009....
Nuclear factor erythroid 2-related factor 2 protects against beta amyloidKatja Kanninen
Department of Neurobiology, AI Virtanen Institute for Molecular Sciences, Kuopio University, Kuopio, Finland
Mol Cell Neurosci 39:302-13. 2008..The findings suggest that the Nrf2-ARE pathway may be impaired in AD and that induction of the Nrf2-ARE defence mechanism may prevent or delay AD-like pathology...
The R6 lines of transgenic mice: a model for screening new therapies for Huntington's diseaseJoana M Gil
Division of Medical Sciences, Island Medical Program, University of Victoria, Victoria, BC, V8W 2Y2, Canada
Brain Res Rev 59:410-31. 2009..Although many of these treatments were beneficial in R6 mice, they may not be as effective in HD patients, and thus the search for a combination of therapies that will rescue the human condition continues...
Survivin: a target from brain cancer to neurodegenerative diseaseSara Baratchi
Centre for Biotechnology and Interdisciplinary Biosciences BioDeakin, Institute for Technology Research and Innovation ITRI, Deakin University, Waurn Ponds, Victoria, Australia
Crit Rev Biochem Mol Biol 45:535-54. 2010..Due to the various roles of survivin during cell division and apoptosis, targeting this protein illustrates a new therapeutic window for the treatment of neurodegenerative diseases...
Intraputamenal infusion of glial cell line-derived neurotrophic factor in PD: a two-year outcome studyNikunj K Patel
Frenchay Hospital, Institute of Neurosciences, Bristol, United Kingdom
Ann Neurol 57:298-302. 2005....
Both systemic and local application of granulocyte-colony stimulating factor (G-CSF) is neuroprotective after retinal ganglion cell axotomyTobias Frank
Department of Neurology, University Medical Center Gottingen, Gottingen, Germany
BMC Neurosci 10:49. 2009..In addition, G-CSF provided neuroprotection in models of neuronal cell death. Here we used the retinal ganglion cell (RGC) axotomy model to compare effects of local and systemic application of neuroprotective molecules...
Inflammatory mechanisms in ischemic stroke: therapeutic approachesShaheen E Lakhan
Global Neuroscience Initiative Foundation, Los Angeles, CA, USA
J Transl Med 7:97. 2009..However, recent studies showing that regulatory T cells are major cerebroprotective immunomodulators after stroke suggest that targeting the endogenous adaptive immune response may offer novel promising neuroprotectant therapies...
Research Grants
- INTERLEUKIN-1 AND PERINATAL BRAIN INJURYFaye Silverstein; Fiscal Year: 1999..of observed effects are to be assessed, as well as effects produced when IL-1ra is combined with other neuroprotective agents such as MK-801...
- New York-Presbyterian NETT ConsortiumStephan Mayer; Fiscal Year: 2007..ischemic stroke, midazolam infusion for refractory status epilepticus, and clinical trials evaluating neuroprotective agents for acute stroke, thrombolytic therapy for intraventricular hemorrhage, and ultra-early hemostatic therapy ..
- Molecular Interventions for Bipolar DisorderALAN PAUL KOZIKOWSKI; Fiscal Year: 2010..the pro-apoptotic properties of the GSK-3 enzyme suggest a potential use of such inhibitors as neuroprotective agents. Neuroprotection may further contribute to the therapeutic efficacy of mood disorder drugs...
- Molecular Interventions for Bipolar DisorderAlan Kozikowski; Fiscal Year: 2007..the pro-apoptotic properties of the GSK-3 enzyme suggest a potential use of such inhibitors as neuroprotective agents. Neuroprotection may further contribute to the therapeutic efficacy of mood disorder drugs...
- Molecular Interventions for Bipolar DisorderAlan Kozikowski; Fiscal Year: 2009..the pro-apoptotic properties of the GSK-3 enzyme suggest a potential use of such inhibitors as neuroprotective agents. Neuroprotection may further contribute to the therapeutic efficacy of mood disorder drugs...
- Stem cell-mediated delivery of neurotrophic factors for treatment of glaucomaDonald S Sakaguchi; Fiscal Year: 2010..is that transplanted, genetically modified bone marrow-derived stem cells can be used as effective neuroprotective agents to mediate preservation and rescue of visual function in the rat model of experimental glaucoma...
- Novel Mitochondrial Targeted Neuroprotectants for GlaucomaLeonard Levin; Fiscal Year: 2007....
- Cerebal Ischemia During Anesthesia and SurgeryPiyush Patel; Fiscal Year: 2004..Anesthetics are logical candidate neuroprotective agents because they reduce excitotoxic injury...
- Parkinson's Disease Neuroprotection Clinical CenterCharles Adler; Fiscal Year: 2005..To this end creating a multi-center study group to run clinical trials of potential neuroprotective agents has been set as a goal of the NIH...
- Insecticide Action at the Local Anesthetic ReceptorDavid M Soderlund; Fiscal Year: 2011..This research will provide new insight into the structure of the local anesthetic receptor and its role in the neurotoxic actions of PTIs. ..
- Insecticide Action at the Local Anesthetic ReceptorDAVID SODERLUND; Fiscal Year: 2009..This research will provide new insight into the structure of the local anesthetic receptor and its role in the neurotoxic actions of PTIs. ..
- Insecticide Action at the Local Anesthetic ReceptorDAVID SODERLUND; Fiscal Year: 2007..This research will provide new insight into the structure of the local anesthetic receptor and its role in the neurotoxic actions of PTIs. ..
- HIGH-THROUGHPUT SCREENING ASSAY FOR NEUROPROTECTIVE AGENTSKarima Ferrani Kile; Fiscal Year: 2007....
- Novel visual outcome measures in optic neuritis and multiple sclerosisLaura Balcer; Fiscal Year: 2007..as new visual outcomes for clinical trials in MS, and in acute ON as a model system for future testing of neuroprotective agents. Specific Aim 2: Determine how new visual outcomes, low-contrast letter acuity and OCT, reflect vision-..
- Canonical Transient Receptor Potential Channels and ExcitotoxicityFang Zheng; Fiscal Year: 2009..However, efforts to develop ionotropic glutamate receptor antagonists as neuroprotective agents have yet to be successful; alternative molecular targets for developing neuroprotective compounds need to ..
- Combination Drug Therapy in Huntington's DiseaseROBERT FERRANTE; Fiscal Year: 2007..compounds or their analogs are available for human use and represent the immediate pipeline of candidate neuroprotective agents for clinical trials in HD...
- Canonical Transient Receptor Potential Channels and ExcitotoxicityFang Zheng; Fiscal Year: 2010..However, efforts to develop ionotropic glutamate receptor antagonists as neuroprotective agents have yet to be successful;alternative molecular targets for developing neuroprotective compounds need to ..
- Phase II Trial of Tiopronin in Aneurysmal Subarachnoid HemorrhageEDWARD SANDER CONNOLLY; Fiscal Year: 2010..This would spark further study that could further explore neuroprotective pre-treatment of cerebral ischemia, and thus help neutralize a major source of morbidity and mortality in this disease process. ..
- A Novel Neuroprotective Approach for IschemiaZhi Gang Jiang; Fiscal Year: 2007..At the end of the phase II period, we expect to submit an IND application to the FDA to use PAN-811 for the treatment of transient ischemic stroke and initiate phase Ib clinical trials. ..
- PARAMEDIC FIELD INITIATION OF MAGNESIUM NEUROPROTECTIVEJeffrey Saver; Fiscal Year: 2003..study will demonstrate the feasibility of performing randomized, controlled clinical trials of promising neuroprotective agents in the field...
- Characterizing Beta Lactams/Neuroprotective Drugs/ALSJeffrey Rothstein; Fiscal Year: 2006..These sequential phases will set the stage for future practical translation towards rational clinical trial design. ..
- Peptidic Ligands for Kappa Opioid ReceptorsJANE ALDRICH; Fiscal Year: 2007..Kappa receptor ligands also have a number of other potential therapeutic applications, including as neuroprotective agents and potentially in the treatment of AIDS...
- A HIGH-THROUGHPUT SCREEN FOR ANTI-NECROTIC COMPOUNDSDONALD KIRSCH; Fiscal Year: 2006..2) Execute a pilot screen of -3000 highly selected compounds to identify neuroprotective agents. A library of known bioactive compounds, including many currently marketed drugs, will be screened for ..
- PARKINSON DISEASE NEUROPROTECTION CLINICAL TRIAL CENTERBala Manyam; Fiscal Year: 2005..abstract_text> ..
- Novel Clinical and Ocular Imaging Outcomes with Long-Term Follow-Up in MSLaura Balcer; Fiscal Year: 2010..in MS clinical trials, particularly for the anticipated next generation of trials that will involve neuroprotective agents. While our cross-sectional, preliminary longitudinal, and clinical trial data represent a significant step ..
- BLOOD/BRAIN BARRIER DRUG DELIVERY OF BDNF IN ISCHEMIAWilliam Pardridge; Fiscal Year: 2002Neurotrophins, such as brain-derived neurotrophic factor (BDNF), are potential neuroprotective agents for the treatment of stroke, trauma, and neurodegenerative diseases...
- Neurotrophin Blood/Brain Barrier Delivery in IschemiaWilliam Pardridge; Fiscal Year: 2006Neurotrophins are powerful neuroprotective agents in global or regional brain ischemia when the protein is injected directly into the ischemic brain...
- Endogenous neuroprotective agents in Parkinson's diseaseAmanda Smith; Fiscal Year: 2007..The mentors that are described herein will actively participate in this undertaking and will further mediate increasing the network of neuroscientists in which I interact locally and nationally. ..
