Research Topics
| W E StumpfSummaryAffiliation: University of North Carolina Country: USA Publications
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Detail Information
Publications
Drugs in the brain--cellular imaging with receptor microscopic autoradiographyWalter E Stumpf
University of North Carolina Chapel Hill, NC 27516, USA
Prog Histochem Cytochem 47:1-26. 2012..New spectrometric methods, like MALDI-MSI, are unlikely to furnish the same information as receptor microautoradiography does, but can provide important correlative molecular information...
In vivo target recognition with high-resolution imaging: significance for drug developmentWalter E Stumpf
University of North Carolina, Chapel Hill, NC, USA
Eur J Drug Metab Pharmacokinet 35:15-22. 2010....
Vitamin D and the digestive systemWalter E Stumpf
University of North Carolina, Chapel Hill, NC, USA
Eur J Drug Metab Pharmacokinet 33:85-100. 2008....
Salivary glands epithelial and myoepithelial cells are major vitamin D targetsWalter E Stumpf
University of North Carolina at Chapel Hill, NC, USA
Eur J Drug Metab Pharmacokinet 32:123-9. 2007....
Skin research and drug localization with receptor microscopic autoradiographyWalter E Stumpf
University of North Carolina at Chapel Hill, NC 27516, USA
Exp Dermatol 17:133-8. 2008..Examples of autoradiograms include in vivo applications of 3H-vitamin D, 3H-OCT (oxacalcitriol), 3H-oestradiol and 3H-retinoic acid. For topical applications, routes of delivery and sites of deposition and retention are demonstrated...
Memo to the FDA and ICH: appeal for in vivo drug target identification and target pharmacokinetics Recommendations for improved procedures and requirementsWalter E Stumpf
2612 Damascus Church Rd, Chapel Hill, NC 27516, USA
Drug Discov Today 12:594-8. 2007..False negatives and false positives of favored 'expedient' procedures allow drugs to reach the market with misleading and inaccurate information about the total drug effect...
Receptor localization of steroid hormones and drugs: discoveries through the use of thaw-mount and dry-mount autoradiographyW E Stumpf
University of North Carolina at Chapel Hill, USA
Braz J Med Biol Res 31:197-206. 1998..Receptor autoradiography with cellular resolution has become an indispensable tool in drug research and development, since information can be obtained that is difficult or impossible to gain otherwise...
The dose makes the medicineWalter E Stumpf
University of North Carolina at Chapel Hill and International Institute of Drug Distribution, Cytopharmacology and Cytotoxicology, 2612 Damascus Church Road, Chapel Hill, NC 27516, USA
Drug Discov Today 11:550-5. 2006..It also allows considerations of systems biology [i.e. integral (gestalt) pharmacology] exemplified by the drug homunculus, as in the case of vitamin D, that might lead to new paradigms and drug design...
Drug localization and targeting with receptor microscopic autoradiographyWalter E Stumpf
University of North Carolina at Chapel Hill, NC, USA
J Pharmacol Toxicol Methods 51:25-40. 2005....
Receptor microscopic autoradiography for the study of percutaneous absorption, in vivo skin penetration, and cellular-intercellular depositionNaohiko Hayakawa
Product Research Department, Chugai Pharmaceutical Co, Ltd, Fuji Gotemba Research Laboratories, 1 135, Komakado, Gotemba, Shizuoka 412 8513, Japan
J Pharmacol Toxicol Methods 50:131-7. 2004..We tested this using (3)H-Maxacalcitol...
Limitations and advantages of whole body autoradiography in the study of tissue distribution of drugs. Response to Dr. SolonWalter E Stumpf
J Pharmacol Toxicol Methods 48:185-6; author reply 187-9. 2002
In vivo time-course of receptor binding in the parathyroid gland of the vitamin D analogue [(3)H]1,25-dihydroxy-22-oxavitamin D(3) compared with [(3)H]1,25-dihydroxyvitamin D(3), determined by micro-autoradiographyNobuo Koike
Fuji Gotemba Laboratories, Chugai Pharmaceutical Co, Ltd, Gotemba, Shizuoka, Japan
Nephrol Dial Transplant 17:53-7. 2002....
Sweat gland epithelial and myoepithelial cells are vitamin D targetsNobuo Koike
Fuji Gotemba Research Laboratories, Chugai Pharmaceutical Company Ltd, Shizuoka, Japan
Exp Dermatol 16:94-7. 2007..The results suggest genomic regulation of cell proliferation and differentiation, as well as of secretory and excretory functions, indicating potential therapies for impaired secretion as in hypohidrosis of aged and diseased skin...
The main role of vitamin D: seasonal regulation of vital functions. High-resolution target recognition leads to a new paradigm and advanced drug developmentWalter E Stumpf
Eur J Drug Metab Pharmacokinet 32:1-6. 2007
Limitations of whole-body autoradiography without receptor microautoradiographyWalter E Stumpf
J Pharmacol Toxicol Methods 48:127-8; author reply 129-30. 2002
Estradiol receptor binding to the epithelium of uterine lumen and glands: region- and time-related changes during preimplantation and periimplantation periods studied by autoradiographyTelma M T Zorn
Laboratory of Biology of Reproduction, Department of Histology and Embryology, Institute of Biomedical Sciences, University of Sao Paulo, 05508 900, Sao Paulo, Brazil
Histochem Cell Biol 120:1-12. 2003..The strong (3)H-estradiol binding to glandular epithelium suggests that estradiol exerts pronounced effects on glandular activities in the periimplantation period...
