Research Topics
Genomes and Genes | Lina YaoSummaryAffiliation: Gilead Sciences Country: USA Publications
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Publications
Inhibition of aldehyde dehydrogenase-2 suppresses cocaine seeking by generating THP, a cocaine use-dependent inhibitor of dopamine synthesisLina Yao
Gilead Sciences, Palo Alto, California, USA
Nat Med 16:1024-8. 2010..Selective inhibition of ALDH-2 may have therapeutic potential for treating human cocaine addiction and preventing relapse...
Nav1.5-dependent persistent Na+ influx activates CaMKII in rat ventricular myocytes and N1325S miceLina Yao
Department of Biology, Gilead Sciences, Palo Alto, California 94304, USA
Am J Physiol Cell Physiol 301:C577-86. 2011..5, further promoting Na(+) influx. Pharmacological inhibition of either CaMKII or Na(v)1.5 can ameliorate cardiac dysfunction caused by excessive Na(+) influx...
Nicotine and ethanol activate protein kinase A synergistically via G(i) betagamma subunits in nucleus accumbens/ventral tegmental cocultures: the role of dopamine D(1)/D(2) and adenosine A(2A) receptorsYuichiro Inoue
Department of Neurology, Ernest Gallo Clinic and Research Center, University of California, San Francisco, California, USA
J Pharmacol Exp Ther 322:23-9. 2007....
Up-regulation of AGS3 during morphine withdrawal promotes cAMP superactivation via adenylyl cyclase 5 and 7 in rat nucleus accumbens/striatal neuronsPeidong Fan
Gilead Sciences, Inc, 3172 Porter Drive, Palo Alto, California 94304, USA
Mol Pharmacol 76:526-33. 2009..Our findings identify a critical role for AC 5 and 7 and A2A receptors for up-regulation of AGS3 in morphine withdrawal-induced cAMP superactivation...
Suppression of heavy drinking and alcohol seeking by a selective ALDH-2 inhibitorMaria P Arolfo
CV Therapeutics, Palo Alto, CA, USA
Alcohol Clin Exp Res 33:1935-44. 2009..However, daidzin can reduce drinking in some rodents without necessarily increasing acetaldehyde. Therefore, a selective ALDH-2 inhibitor might affect other metabolic factors involved in regulating drinking...
Characterization of the potency, selectivity, and pharmacokinetic profile for six adenosine A2A receptor antagonistsMing Yang
Department of Pharmacology, CV Therapeutics, Inc, Palo Alto, CA 94304, USA
Naunyn Schmiedebergs Arch Pharmacol 375:133-44. 2007..Among the six A2A-antagonists, KW-6002 is the best for use in in vivo animal studies, particularly for a CNS target, based on its bioavailability, half life, and brain penetration...
Dopamine and ethanol cause translocation of epsilonPKC associated with epsilonRACK: cross-talk between cAMP-dependent protein kinase A and protein kinase C signaling pathwaysLina Yao
CV Therapeutics, Inc, 3172 Porter Drive, Palo Alto, CA 94304, USA
Mol Pharmacol 73:1105-12. 2008..PKA and PKC signaling have been implicated in alcohol rewarding properties in the mesolimbic dopamine system. Cross-talk between PKA and PKC may underlie some of the behaviors associated with alcoholism...
Ambrisentan and tadalafil synergistically relax endothelin-induced contraction of rat pulmonary arteriesFaquan Liang
Department of Biology, Gilead Sciences, Inc, 1651 Page Mill Rd, Palo Alto, CA 94304, USA
Hypertension 59:705-11. 2012....
Adenosine A2a blockade prevents synergy between mu-opiate and cannabinoid CB1 receptors and eliminates heroin-seeking behavior in addicted ratsLina Yao
CV Therapeutics, Inc, 3172 Porter Drive, Palo Alto, CA 94304, USA
Proc Natl Acad Sci U S A 103:7877-82. 2006..These findings suggest that A2a antagonists might be effective therapeutic agents in the management of abstinent heroin addicts...
