Research Topics
Genomes and Genes | I HersSummaryAffiliation: University of Bristol Country: UK Publications
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Publications
The protein kinase C inhibitors bisindolylmaleimide I (GF 109203x) and IX (Ro 31-8220) are potent inhibitors of glycogen synthase kinase-3 activityI Hers
Department of Biochemistry, School of Medical Sciences, University of Bristol, UK
FEBS Lett 460:433-6. 1999..We propose that bisindolylmaleimide I and IX can directly inhibit GSK-3, and that this may explain some of the previously reported insulin-like effects on glycogen synthase activity...
Insulin-like growth factor-1 potentiates platelet activation via the IRS/PI3Kalpha pathwayIngeborg Hers
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol, UK
Blood 110:4243-52. 2007..These results demonstrate that IGF-1 activates the IGF receptor/IRS/PI3K/PKB pathway, and that PI3Kalpha is essential for the potentiatory effect of IGF-1 on platelet responses...
Identification of p122RhoGAP (deleted in liver cancer-1) Serine 322 as a substrate for protein kinase B and ribosomal S6 kinase in insulin-stimulated cellsIngeborg Hers
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol BS8 1TD, United Kingdom
J Biol Chem 281:4762-70. 2006..These results demonstrate that p122RhoGAP Ser-322 acts as an integrator of signal transduction in a manner dependent on the cellular context...
Mechanism of feedback regulation of insulin receptor substrate-1 phosphorylation in primary adipocytesIngeborg Hers
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol BS8 1TD, UK
Biochem J 388:713-20. 2005....
Reciprocal feedback regulation of insulin receptor and insulin receptor substrate tyrosine phosphorylation by phosphoinositide 3-kinase in primary adipocytesIngeborg Hers
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol BS8 1TD, UK
Biochem J 368:875-84. 2002....
Protein kinase B phosphorylation of PIKfyve regulates the trafficking of GLUT4 vesiclesDaniel C Berwick
Department of Biochemistry, School of Medical Sciences, University of Bristol, University Walk, Bristol, BS8 1TD, UK
J Cell Sci 117:5985-93. 2004....
Insulin/IGF-1 hybrid receptor expression on human platelets: consequences for the effect of insulin on platelet functionR W Hunter
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol, UK
J Thromb Haemost 7:2123-30. 2009..This study investigated the possibility that platelets express hybrid receptors, which may affect insulin action on platelet function...
Protein kinase C-mediated phosphorylation and activation of PDE3A regulate cAMP levels in human plateletsRoger W Hunter
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol BS8 1TD, UK
J Biol Chem 284:12339-48. 2009....
The identification of ATP-citrate lyase as a protein kinase B (Akt) substrate in primary adipocytesDaniel C Berwick
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol BS8 1TD, United Kingdom
J Biol Chem 277:33895-900. 2002..Taken together, these results demonstrate that serine 454 of ATP-citrate lyase is a novel and major in vivo substrate for protein kinase B...
PKC-interacting proteins: from function to pharmacologyAlastair W Poole
Department of Pharmacology, School of Medical Sciences, University Walk, Bristol BS8 1TD, UK
Trends Pharmacol Sci 25:528-35. 2004..In this article, we review recent work on C-KIPs and the implications for pharmacological and therapeutic development...
The PKB inhibitor Akti-1/2 potentiates PAR-1-mediated platelet function independently of its ability to block PKBR W Hunter
Department of Biochemistry, School of Medicine Sciences, University of Bristol, Bristol, UK
J Thromb Haemost 6:1923-32. 2008..Recently, a selective, non-ATP-competitive PKB inhibitor, Akti-1/2 has been reported, but the efficacy and specificity against PKB activation in platelet function is unknown...
Regulation of small GTP-binding proteins by insulinG I Welsh
Department of Biochemistry, School of Medical Sciences, University of Bristol, Bristol BS8 ITD, UK
Biochem Soc Trans 34:209-12. 2006..We review recent evidence that this may be the case, and place specific emphasis on the role of these pathways in insulin-stimulated glucose uptake...
Understanding the therapeutic action of recombinant factor VIIa in platelet disordersIngeborg Hers
Department of Biochemistry, School of Medical Sciences, University of Bristol, University Walk, Bristol BS8 1TD, UK
Platelets 19:571-81. 2008..This review summarizes the clinical and experimental evidence supporting a potentiating effect of FVIIa on platelet activation and discusses the likely mechanism of action...
