T Kenakin

Summary

Publications

  1. ncbi Efficacy in drug receptor theory: outdated concept or under-valued tool?
    T Kenakin
    Department of Receptor Biochemistry, Glaxo Wellcome Research and Development, Research Triangle Park, NC 27709, USA
    Trends Pharmacol Sci 20:400-5. 1999
  2. ncbi Inverse, protean, and ligand-selective agonism: matters of receptor conformation
    T Kenakin
    Department of Receptor Biochemistry, Glaxo SmithKline Research and Development, Research Triangle Park, North Carolina 27709, USA
    FASEB J 15:598-611. 2001

Detail Information

Publications2

  1. ncbi Efficacy in drug receptor theory: outdated concept or under-valued tool?
    T Kenakin
    Department of Receptor Biochemistry, Glaxo Wellcome Research and Development, Research Triangle Park, NC 27709, USA
    Trends Pharmacol Sci 20:400-5. 1999
    ....
  2. ncbi Inverse, protean, and ligand-selective agonism: matters of receptor conformation
    T Kenakin
    Department of Receptor Biochemistry, Glaxo SmithKline Research and Development, Research Triangle Park, North Carolina 27709, USA
    FASEB J 15:598-611. 2001
    ..This paper reviews evidence for the existence of the various types of agonism and the potential therapeutic utility of different agonist types.-Kenakin, T. Inverse, protean, and ligand-selective agonism: matters of receptor conformation...