Research Topics
Species | Tomohiro NabekuraSummaryCountry: Japan Publications
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Publications
Overcoming multidrug resistance in human cancer cells by natural compoundsTomohiro Nabekura
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Higashi jima, Akiha ku, Niigata 956 8603, Japan
Toxins (Basel) 2:1207-24. 2010..In this review, studies on the effects of natural compounds on P-glycoprotein and anticancer drug efflux transporters are summarized...
Inhibition of anticancer drug efflux transporter P-glycoprotein by rosemary phytochemicalsTomohiro Nabekura
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Higashi jima, Akiha ku, Niigata 956 8603, Japan
Pharmacol Res 61:259-63. 2010..These results suggest that rosemary phytochemicals, such as carnosic acid, have inhibitory effects on anticancer drug efflux transporter P-glycoprotein and may become useful to enhance the efficacy of cancer chemotherapy...
Effects of chemopreventive citrus phytochemicals on human P-glycoprotein and multidrug resistance protein 1Tomohiro Nabekura
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Niigata, Japan
Eur J Pharmacol 600:45-9. 2008..These results suggest that chemopreventive citrus phytochemicals, such as nobiletin found in oranges, have inhibitory effects on P-glycoprotein and/or MRP1, and may cause food-drug interactions...
Inhibition of P-glycoprotein and multidrug resistance protein 1 by dietary phytochemicalsTomohiro Nabekura
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Higashi jima, Akiha ku, Niigata 956 8603, Japan
Cancer Chemother Pharmacol 62:867-73. 2008....
Effect of triterpenoids isolated from the floral spikes of Betula platyphylla var. japonica on P-glycoprotein functionMichiko Sekiya
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Niigata, Japan
Planta Med 73:1558-62. 2007..In addition, compounds 13 and 20 showed a weak inhibitory activity of P-gp ATPase. These results suggested that MDR reversing effects of compounds 13 and 20 are partly involved in inhibition of P-gp ATPase...
Enhanced skin permeation of diclofenac by ion-pair formation and further enhancement by microemulsionMohammad Abu Hena Mostofa Kamal
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Niigata, Japan
Chem Pharm Bull (Tokyo) 55:368-71. 2007..The present findings suggest the usefulness of combined use of ion-pairs with microemulsions for enhancement of skin permeation of ionic drugs...
Structure-activity relationships of the inhibitory effects of flavonoids on P-glycoprotein-mediated transport in KB-C2 cellsShuji Kitagawa
Niigata University of Pharmacy and Applied Life Sciences, Japan
Biol Pharm Bull 28:2274-8. 2005..These results suggested that hydrophobicity as well as planar structure is important for the inhibitory effects of flavonoids on P-gp-mediated transport...
Effects of dietary chemopreventive phytochemicals on P-glycoprotein functionTomohiro Nabekura
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Niigata, Japan
Biochem Biophys Res Commun 327:866-70. 2005..These results suggest that dietary phytochemicals, such as capsaicin, curcumin, [6]-gingerol, and resveratrol, have inhibitory effects on P-glycoprotein and potencies to cause drug-food interactions...
Effects of plant sterols on human multidrug transporters ABCB1 and ABCC1Tomohiro Nabekura
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Higashi jima, Akiha ku, Niigata 956 8603, Japan
Biochem Biophys Res Commun 369:363-8. 2008..These results suggest that guggulsterone, a natural dietary hypolipidemic agent have dual inhibitory effects on P-gp and MRP1 and the potencies to cause food-drug interactions...
Effects of alkyl gallates on P-glycoprotein functionShuji Kitagawa
Laboratory of Pharmaceutics, Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Japan
Biochem Pharmacol 70:1262-6. 2005..The cytotoxicity of daunorubicin was recovered in the presence of alkyl gallates possibly due to their inhibition of P-gp function...
Inhibition of P-glycoprotein function by tea catechins in KB-C2 cellsShuji Kitagawa
Niigata University of Pharmacy and Applied Life Sciences, Kamishin ei cho 5 13 2, 950 2081, Japan
J Pharm Pharmacol 56:1001-5. 2004....
Enhanced skin permeation of salicylate by ion-pair formation in non-aqueous vehicle and further enhancement by ethanol and l-mentholMohammad Abu Hena Mostofa Kamal
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Japan
Chem Pharm Bull (Tokyo) 54:481-4. 2006....
Permeability of ionized salicylate derivatives through guinea pig dorsal skinMohammad Abu Hena Mostofa Kamal
Faculty of Pharmaceutical Sciences, Niigata University of Pharmacy and Applied Life Sciences, Niigata, Japan
Chem Pharm Bull (Tokyo) 53:441-3. 2005..These findings suggested that the ionic permeation pathway of salicylate derivatives is controlled by hydrophobic as well as hydrophilic properties...
