Galli U, Ciraolo E, Massarotti A, Margaria J, Sorba G, Hirsch E, et al
. The Guareschi Pyridine Scaffold as a Valuable Platform for the Identification of Selective PI3K Inhibitors. Molecules. 2015;20:17275-87 pubmed publisher
..Compound 9b is a selective inhibitor against the PI3KÎ± isoform, maintaining a good inhibitory activity. Docking studies were also performed in order to rationalize its profile of selectivity. ..