Research Topics
| Robert J KindersSummaryAffiliation: National Institutes of Health Country: USA Publications
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Detail Information
Publications
Preclinical modeling of a phase 0 clinical trial: qualification of a pharmacodynamic assay of poly (ADP-ribose) polymerase in tumor biopsies of mouse xenograftsRobert J Kinders
Laboratory of Human Toxicology and Pharmacology, Applied Developmental Research Support Directorate, Science Applications International Corporation Frederick, Inc, National Cancer Institute Frederick, Frederick, MD 21702, USA
Clin Cancer Res 14:6877-85. 2008..S. Food and Drug Administration's Exploratory Investigational New Drug Application. Performance of the study design, needle biopsy procedure, and validated pharmacodynamic assay were evaluated in human tumor xenograft models...
Development of a validated immunofluorescence assay for ?H2AX as a pharmacodynamic marker of topoisomerase I inhibitor activityRobert J Kinders
Laboratory of Human Toxicology and Pharmacology, Applied Developmental Research Support Directorate, Science Applications International Corporation Frederick, Inc, NationalCancer Institute Frederick, Frederick, MD 21702, USA
Clin Cancer Res 16:5447-57. 2010..A quantitative pharmacodynamic immunofluorescence assay for ?H2AX was developed, validated, and tested in human tumor xenograft models with the use of clinically relevant procedures...
Monitoring drug-induced gammaH2AX as a pharmacodynamic biomarker in individual circulating tumor cellsLihua H Wang
Laboratory of Human Toxicology and Pharmacology, Science Applications International Corporation, Frederick, MD, USA
Clin Cancer Res 16:1073-84. 2010..Here, we describe an assay that directly examines changes in levels of the nuclear DNA damage marker gammaH2AX in individual CTCs of patients treated with chemotherapeutic agents...
Increased antitumor activity of bevacizumab in combination with hypoxia inducible factor-1 inhibitionAnnamaria Rapisarda
SAIC Frederick Inc, National Cancer Institue at Frederick, Frederick, MD 21702, USA
Mol Cancer Ther 8:1867-77. 2009..These results strongly suggest that combination of anti-vascular endothelial growth factor antibodies with HIF-1 inhibitors is an attractive therapeutic strategy targeting in the hypoxic tumor microenvironment...
Topoisomerase I levels in the NCI-60 cancer cell line panel determined by validated ELISA and microarray analysis and correlation with indenoisoquinoline sensitivityThomas D Pfister
Laboratory of Human Toxicology and Pharmacology, Applied Developmental Research Support Directorate, Science Applications International Corporation Frederick Inc, National Cancer Institute Frederick, Frederick, MD 21702, USA
Mol Cancer Ther 8:1878-84. 2009....
