Research Topics
Species | Rudi BaoSummaryAffiliation: Curis Inc Country: USA Publications
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Detail Information
Publications
CUDC-305, a novel synthetic HSP90 inhibitor with unique pharmacologic properties for cancer therapyRudi Bao
Curis, Inc, Cambridge, Massachusetts 02138, USA
Clin Cancer Res 15:4046-57. 2009..We designed and synthesized CUDC-305, an HSP90 inhibitor of the novel imidazopyridine class. Here, we report its unique pharmacologic properties and antitumor activities in a variety of tumor types...
Targeting heat shock protein 90 with CUDC-305 overcomes erlotinib resistance in non-small cell lung cancerRudi Bao
Oncology, Curis, Inc, 45 Moulton Street, Cambridge, MA 02138, USA
Mol Cancer Ther 8:3296-306. 2009..These results suggest that CUDC-305 holds promise for the treatment of NSCLC with primary or acquired resistance to EGFR inhibitor therapy...
Discovery of 7-(4-(3-ethynylphenylamino)-7-methoxyquinazolin-6-yloxy)-N-hydroxyheptanamide (CUDc-101) as a potent multi-acting HDAC, EGFR, and HER2 inhibitor for the treatment of cancerXiong Cai
Curis Inc, 45 Moulton Street, Cambridge, Massachusetts 02138, USA
J Med Chem 53:2000-9. 2010....
CUDC-101, a multitargeted inhibitor of histone deacetylase, epidermal growth factor receptor, and human epidermal growth factor receptor 2, exerts potent anticancer activityCheng Jung Lai
Curis, Inc, Cambridge, Massachusetts, USA
Cancer Res 70:3647-56. 2010..Cancer Res; 70(9); 3647-56. (c)2010 AACR...
