Research Topics
Genomes and Genes | Herbert M PinedoSummaryAffiliation: VU University Medical Center Country: The Netherlands Publications
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Publications
Thrombosis, prevalence and new evidence on current perceptions of riskHerbert M Pinedo
Department of Medical Oncology, Free University of Amsterdam, P O Box 7057, 1007 MB, Amsterdam, The Netherlands
Cancer Treat Rev 29:3-5. 2003..Most clinicians treating medical (non-surgical) cancer patients perceived pancreatic tumours to carry a high thrombosis risk in the absence of thromboprophylaxis...
Extended neoadjuvant chemotherapy in locally advanced breast cancer combined with GM-CSF: effect on tumour-draining lymph node dendritic cellsH M Pinedo
Department of Medical Oncology, VU University Medical Center, PO Box 7057, 1007 MB Amsterdam, The Netherlands
Eur J Cancer 39:1061-7. 2003....
Pronounced antitumor efficacy by extracellular activation of a doxorubicin-glucuronide prodrug after adenoviral vector-mediated expression of a human antibody-enzyme fusion proteinMichelle de Graaf
Department of Medical Oncology, Division of Gene Therapy, VU University Medical Center, 1007 MB Amsterdam, The Netherlands
Hum Gene Ther 15:229-38. 2004..1 days (p < 0.01), while virus alone had no effect. Thus, we have successfully shown that an adenovirus vector encoding a secreted, targeted form of human beta-glucuronidase can further improve DOX-GA3 monotherapy...
Evidence for a role of p38 kinase in hypoxia-inducible factor 1-independent induction of vascular endothelial growth factor expression by sodium arseniteMonique C A Duyndam
Department of Medical Oncology, Vrije Universiteit Medical Center, Amsterdam 1081 HV, The Netherlands
J Biol Chem 278:6885-95. 2003..Altogether, these data suggest that not HIF-1, but rather p38, mediates induction of VEGF mRNA expression by sodium arsenite...
Conditionally replicative adenovirus with tropism expanded towards integrins inhibits osteosarcoma tumor growth in vitro and in vivoAdhiambo M Witlox
Department of Orthopedic Surgery, VU University Medical Center, Amsterdam, The Netherlands
Clin Cancer Res 10:61-7. 2004..CONCLUSIONS: Targeting adenovirus toward integrins rendered OS cells more sensitive to killing by Ad5-Delta24RGD. These findings suggest that Ad5-Delta24RGD has potential for use in OS treatment...
The activity profile of the hexacyclic camptothecin derivative DX-8951f in experimental human colon cancer and ovarian cancerAnnemarie H van Hattum
Department of Medical Oncology, Vrije Universiteit Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
Biochem Pharmacol 64:1267-77. 2002..Addition of cisplatin or paclitaxel improved the in vivo antitumor effects of DX-8951f...
Prolonged maturation and enhanced transduction of dendritic cells migrated from human skin explants after in situ delivery of CD40-targeted adenoviral vectorsTanja D de Gruijl
Division of Immunotherapy, Department of Medical Oncology, Vrije Universiteit University Medical Center, Amsterdam, The Netherlands
J Immunol 169:5322-31. 2002..Because DC targeting in vivo might obviate the need for the in vitro culture of autologous DC for adoptive transfer, CD40-targeted Ad vectors constitute a promising new vaccine modality for tumor immunotherapy...
Reduced growth, increased vascular area, and reduced response to cisplatin in CD13-overexpressing human ovarian cancer xenograftsYvette van Hensbergen
Department of Medical Oncology, , 1007 MB Amsterdam, The Netherlands
Clin Cancer Res 10:1180-91. 2004..Further elucidation of the mechanism of the observed effects of CD13 is warranted to better understand its role in the pathophysiology of ovarian cancer...
A postmigrational switch among skin-derived dendritic cells to a macrophage-like phenotype is predetermined by the intracutaneous cytokine balanceTanja D de Gruijl
Department of Medical Oncology, Division of Immunotherapy, VU University Medical Center, Amsterdam, The Netherlands
J Immunol 176:7232-42. 2006....
The organotypic multicellular spheroid is a relevant three-dimensional model to study adenovirus replication and penetration in human tumors in vitroJacques Grill
Division of Gene Therapy, Department of Medical Oncology, VU University Medical Center, Amsterdam, The Netherlands
Mol Ther 6:609-14. 2002..We can conclude that organotypic spheroids offer a versatile in vitro system for studying distribution, spread, and oncolysis by adenoviruses in a clinically relevant model...
Polarization of Valpha24+ Vbeta11+ natural killer T cells of healthy volunteers and cancer patients using alpha-galactosylceramide-loaded and environmentally instructed dendritic cellsHans J J van der Vliet
Department of Medical Oncology, Vrije Universiteit Medisch Centrum, Amsterdam, The Netherlands
Cancer Res 63:4101-6. 2003....
Gene-directed enzyme prodrug therapy for osteosarcoma: sensitization to CPT-11 in vitro and in vivo by adenoviral delivery of a gene encoding secreted carboxylesterase-2Dinja Oosterhoff
Division of Gene Therapy, Department of Medical Oncology, VU University Medical Center, 1007 MB, Amsterdam, The Netherlands
Mol Cancer Ther 2:765-71. 2003..05). Taken together, these data suggest that OS cells are sensitive for the combination of Ad-sCE2 and CPT-11...
A CD34(+) human cell line model of myeloid dendritic cell differentiation: evidence for a CD14(+)CD11b(+) Langerhans cell precursorSaskia J A M Santegoets
VU University Medical Center, De Boelelaan 1117, Amsterdam 1081HV, The Netherlands
J Leukoc Biol 80:1337-44. 2006..We conclude that the MUTZ-3 cell line provides a ready and continuous supply of common myeloid precursors, which should facilitate further study of the ontogeny of myeloid DC lineages...
Potential of the conditionally replicative adenovirus Ad5-Delta24RGD in the treatment of malignant gliomas and its enhanced effect with radiotherapyMartine L M Lamfers
Department of Neurosurgery, VU University Medical Center, 1007 MB Amsterdam, The Netherlands
Cancer Res 62:5736-42. 2002..These results support further development of Ad5-Delta24RGD in combination with radiation therapy for treatment of these highly malignant tumors...
A methylester of the glucuronide prodrug DOX-GA3 for improvement of tumor-selective chemotherapyMichelle de Graaf
Department of Medical Oncology, VU University Medical Center, P.O. Box 7057, 1007 MB Amsterdam, The Netherlands
Biochem Pharmacol 68:2273-81. 2004..This effect may even be more pronounced in man, because of the lower plasma esterase activity than measured in mice...
MUTZ-3, a human cell line model for the cytokine-induced differentiation of dendritic cells from CD34+ precursorsAllan J Masterson
Department of Medical Oncology, Division Immunotherapy, VU University Medical Center VUmc, Amsterdam, The Netherlands
Blood 100:701-3. 2002..These findings demonstrate the unique suitability of MUTZ-3 cells as an unlimited source of CD34+ DC progenitors for the study of cytokine-induced DC differentiation...
O6-methylguanine-DNA-methyltransferase promoter demethylation is involved in basic fibroblast growth factor induced resistance against temozolomide in human melanoma cellsDennis Fontijn
Department of Medical Oncology, VU University Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
Mol Cancer Ther 6:2807-15. 2007..There were no changes in sensitivity to docetaxel and doxorubicin. In conclusion, bFGF overexpression can result in resistance against temozolomide mediated by demethylation of the O6-methylguanine-DNA-methyltransferase promoter...
The immunoregulatory role of CD1d-restricted natural killer T cells in diseaseHans J J van der Vliet
The Departments of Pathology, Vrije Universiteit Medisch Centrum, Amsterdam, The Netherlands
Clin Immunol 112:8-23. 2004..Here, we review the immunoregulatory role of NKT cells in disease and discuss NKT cell based immunotherapeutic strategies...
18F-2-fluoro-2-deoxy-d-glucose positron emission tomography in staging of locally advanced breast cancerJacobus J M van Der Hoeven
Departments of Nuclear Medicine and PET Research, Vrije Universiteit University Medical Center, Amsterdam, The Netherlands
J Clin Oncol 22:1253-9. 2004..To prospectively evaluate the effect of adding whole-body (18)F-2-fluoro-2-deoxy-d-glucose (FDG) positron emission tomography (PET) to conventional screening for distant metastases in patients with locally advanced breast cancer (LABC)...
Polymorphisms in the enhancer region of the thymidylate synthase gene are associated with thymidylate synthase levels in normal tissues but not in malignant tissues of patients with colorectal cancerRobert Mauritz
Department of Medical Oncology, VU University Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
Clin Colorectal Cancer 8:146-54. 2009....
Dynamics of antifolate transport via the reduced folate carrier and the membrane folate receptor in murine leukaemia cells in vitro and in vivoRobert Mauritz
Department of Medical Oncology, VU University Medical Center, P O Box 7057, 1007 MB, Amsterdam, The Netherlands
Cancer Chemother Pharmacol 62:937-48. 2008..Collectively, this study underscores that modulation of dietary folate status can provide a basis within which the therapeutic effect of antifolates may be further improved...
Early apoptosis largely accounts for functional impairment of CD34+ cells in frozen-thawed stem cell graftsFransien de Boer
Department of Hematology, VU University Medical Center, 1081 HV Amsterdam, The Netherlands
J Hematother Stem Cell Res 11:951-63. 2002..Further development of this assay should allow its incorporation into the routine CD34(+) assessment of post-thawed samples in clinical flow cytometry laboratories...
Gene therapy for meningioma: improved gene delivery with targeted adenovirusesClemens M F Dirven
Department of Neurosurgery, Vrije Universiteit Medical Center, Amsterdam, The Netherlands
J Neurosurg 97:441-9. 2002..Gene therapy is an emerging strategy for the treatment of brain tumors, which the authors investigated to determine whether adenoviruses could be used for gene transfer in meningioma cells...
A phase I study of the natural killer T-cell ligand alpha-galactosylceramide (KRN7000) in patients with solid tumorsGiuseppe Giaccone
Department of Medical Oncology, Vrije Universiteit Medical Center, HV 1081 Amsterdam, The Netherlands
Clin Cancer Res 8:3702-9. 2002..We performed a dose escalation study of KRN7000 in advanced cancer patients...
Cisplatin and doxorubicin repress Vascular Endothelial Growth Factor expression and differentially down-regulate Hypoxia-inducible Factor I activity in human ovarian cancer cellsMonique C A Duyndam
Department of Medical Oncology, VU University Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
Biochem Pharmacol 74:191-201. 2007..This knowledge may be useful for future treatment schedules including agents that target the HIF-1 signalling pathway...
The 18 kDa isoform of basic fibroblast growth factor is sufficient to stimulate human melanoma growth and angiogenesisDennis Fontijn
Department of Medical Oncology, VU University Medical Center, Amsterdam, The Netherlands
Melanoma Res 17:155-68. 2007..Taken together, overexpression of the 18 kDa basic fibroblast growth factor protein only can promote autocrine melanoma cell growth and paracrine-driven angiogenesis...
Induction of p53 up-regulated modulator of apoptosis messenger RNA by chemotherapeutic treatment of locally advanced breast cancerRutger Middelburg
Department of Medical Oncology, VU University Medical Center, 1007 MB Amsterdam, The Netherlands
Clin Cancer Res 11:1863-9. 2005..Because PUMA is a known member of the family of BH3-only proapoptotic proteins, this finding suggests PUMA's potential importance for the response to anticancer drugs...
Levels of hypoxia-inducible factor-1alpha independently predict prognosis in patients with lymph node negative breast carcinomaReinhard Bos
Department of Pathology, VU University Medical Center, Amsterdam, The Netherlands
Cancer 97:1573-81. 2003..Therefore, the use of immunohistochemical assessment of HIF-1alpha as a new predictor of poor outcome may improve clinical decision-making regarding adjuvant treatment of patients with lymph node negative breast carcinoma...
Protein expression of B-cell lymphoma gene 6 (BCL-6) in invasive breast cancer is associated with cyclin D1 and hypoxia-inducible factor-1alpha (HIF-1alpha)Reinhard Bos
Department of Pathology, VU University Medical Center, Amsterdam, The Netherlands
Oncogene 22:8948-51. 2003..The cases with amplification in BCL-6 showed an increased (25%) incidence of BCL-6 protein overexpression. Thus, this study is the first to show that BCL-6 oncogene activation plays a role in cancers other than lymphomas...
Sulfasalazine down-regulates the expression of the angiogenic factors platelet-derived endothelial cell growth factor/thymidine phosphorylase and interleukin-8 in human monocytic-macrophage THP1 and U937 cellsMichiel de Bruin
Department of Medical Oncology, VU University Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
Mol Pharmacol 66:1054-60. 2004..However, this may also negatively affect capecitabine efficacy...
Thymidylate synthase and dihydropyrimidine dehydrogenase mRNA expression after administration of 5-fluorouracil to patients with colorectal cancerRobert Mauritz
Department of Medical Oncology, VU University Medical Center, Amsterdam, The Netherlands
Int J Cancer 120:2609-12. 2007..2-fold lower than in 18 primary tumors of unexposed patients (p = 0.027). In conclusion, administration of 5FU in vivo influences the gene expression of TS and DPD...
Effects of gemcitabine on cis-platinum-DNA adduct formation and repair in a panel of gemcitabine and cisplatin-sensitive or -resistant human ovarian cancer cell linesGodefridus J Peters
Department of Medical Oncology, VU University Medical Center, 1007 MB Amsterdam, The Netherlands
Int J Oncol 28:237-44. 2006..6-fold directly after exposure but did not clearly affect the AUA0-25 h. In conclusion, dFdC can affect both Pt-DNA adduct formation and repair, depending on the initial sensitivity of the cells...
Neoadjuvant chemoimmunotherapy in locally advanced breast cancer: a new avenue to be exploredJan Buter
Department of Medical Oncology, VU University Medical Center, PO Box 7057, 1007 MB Amsterdam, The Netherlands
Curr Oncol Rep 5:171-6. 2003
Conditionally replicative adenovirus expressing p53 exhibits enhanced oncolytic potencyVictor W van Beusechem
Division of Gene Therapy, Department of Medical Oncology, VU University Medical Center, 1081 HV Amsterdam, The Netherlands
Cancer Res 62:6165-71. 2002..CRAd potency was increased up to >100-fold by p53 expression. We conclude that CRAds expressing p53 are promising new agents for more effective treatment of many human cancers...
Whole-cell cancer vaccination: from autologous to allogeneic tumor- and dendritic cell-based vaccinesTanja D de Gruijl
Department of Medical Oncology, Vrije Universiteit Medical Center, Amsterdam, The Netherlands
Cancer Immunol Immunother 57:1569-77. 2008....
Cytosolic beta-glycosidases for activation of glycoside prodrugs of daunorubicinMichelle de Graaf
Department of Medical Oncology, Vrije Universiteit Medical Center, P.O. Box 7057, 1007 MB Amsterdam, The Netherlands
Biochem Pharmacol 65:1875-81. 2003....
Simulation model of doxorubicin activity in islets of human breast cancer cellsJan Lankelma
Department of Medical Oncology, VU Medical Center, Room BR232, P O Box 7057, 1007 MB Amsterdam, The Netherlands
Biochim Biophys Acta 1622:169-78. 2003..In the model doxorubicin exposure resulted in less cell damage inside the tumor islets than at the rim...
Pretreatment deoxycytidine kinase levels predict in vivo gemcitabine sensitivityJudith R Kroep
Department of Medical Oncology, VU University Medical Center, Amsterdam, The Netherlands
Mol Cancer Ther 1:371-6. 2002..In conclusion, the clear correlation between dCK levels and gemcitabine sensitivity in various murine tumors and human tumor xenografts may be a prognostic parameter when considering gemcitabine therapy...
Beta-glucuronidase-mediated drug releaseMichelle de Graaf
Department of Medical Oncology, Division of Gene Therapy, Vrije Universiteit Medical Centre, P.O. Box 7057, Amsterdam, 1007 MB, The Netherlands
Curr Pharm Des 8:1391-403. 2002..Enhancement of the therapeutic effects of glucuronide prodrugs, also in patients with small tumour lesions, may possibly be achieved by techniques that target beta-glucuronidase specifically to the site of the tumour...
Novel camptothecin derivative BNP1350 in experimental human ovarian cancer: determination of efficacy and possible mechanisms of resistanceAnnemarie H van Hattum
Department of Medical Oncology, Vrije Universiteit Medical Center, Amsterdam, The Netherlands
Int J Cancer 100:22-9. 2002..In contrast to topotecan, BNP1350 proved not to be a good substrate for BCRP. Overall, we conclude that BNP1350 offers advantages over topotecan expressed by high efficacy in experimental human ovarian cancer and poor affinity for BCRP...
Dose-finding study of the multitargeted tyrosine kinase inhibitor SU6668 in patients with advanced malignanciesBart C Kuenen
Department of Medical Oncology, VU Medical Center, Amsterdam, Netherlands
Clin Cancer Res 11:6240-6. 2005..CONCLUSIONS: The maximum tolerated dose of SU6668 given orally, thrice daily under fed conditions, is 100 mg/m2. Because of the low plasma levels reached at this dose level, the efficacy of SU6668 as a single agent is not to be expected...
Homing and clonogenic outgrowth of CD34(+) peripheral blood stem cells: a role for L-selectin?Fransien de Boer
Department of Hematology, VU University Medical Center, Amsterdam, The Netherlands
Exp Hematol 30:590-7. 2002..In the present study, we determined the role of L-selectin in different engraftment steps, i.e., adhesion to endothelial cells, migration, and clonogenic outgrowth by in vitro assays that closely mimic the in vivo situation...
Soluble aminopeptidase N/CD13 in malignant and nonmalignant effusions and intratumoral fluidYvette van Hensbergen
Vrye Universiteit Medical Center, Department of Medical Oncology, 1081 HV Amsterdam, The Netherlands
Clin Cancer Res 8:3747-54. 2002..If so, sCD13 could be a convenient potential marker for tumor load and/or activated tumor endothelium...
On our way to targeted therapy for cachexia in cancer?Manon S A Boddaert
Department of Medical Oncology, VUMC Cancer Center Amsterdam, Amsterdam, The Netherlands
Curr Opin Oncol 18:335-40. 2006..Despite extensive research in an attempt to better understand the mechanisms involved, progress in the management of cancer cachexia has been slow...
Positron emission tomography using 2-deoxy-2-[18F]-fluoro-D-glucose for response monitoring in locally advanced gastroesophageal cancer; a comparison of different analytical methodsJudith R Kroep
Department of Medical Oncology, Amsterdam, The Netherlands
Mol Imaging Biol 5:337-46. 2003..CONCLUSIONS: FDG-PET reliably predicted response in LAGEC. FDG-PET measurements using Patlak analysis or the more clinical applicable SKM and SUV-BW were acceptable alternatives to NLR...
Making use of the primary tumourArnold Baars
Department of Medical Oncology, Vrije Universiteit Medical Centre, Amsterdam, The Netherlands
Bioessays 25:79-86. 2003....
Prostanoids play a major role in the primary tumor-induced inhibition of dendritic cell differentiationClaudia C Sombroek
Department of Pathology, Vrije Universiteit Medical Center, Amsterdam, The Netherlands
J Immunol 168:4333-43. 2002..In conclusion, this study demonstrates that primary tumors negatively impact DC development and function through COX-1 and -2 regulated factors, whereas tumor-derived cell lines may lose this ability upon in vitro propagation...
The effect of fluoropyrimidines with or without thymidine phosphorylase inhibitor on the expression of thymidine phosphorylaseMichiel de Bruin
Department of Medical Oncology, VU University Medical Center, De Boelelaan 1117, P.O. Box 7057, 1081 HV Amsterdam, The Netherlands
Eur J Pharmacol 491:93-9. 2004..This demonstrated that regulation is drug and cell line dependent...
Natural Killer T cellsHans J J van der Vliet
Lancet Oncol 3:574. 2002
Expression of scFvs and scFv fusion proteins in eukaryotic cellsMichelle de Graaf
Division of Gene Therapy, Department of Medical Oncology, Vrije University, Amsterdam, The Netherlands
Methods Mol Biol 178:379-87. 2002
Molecular tests for colorectal cancer screeningLinda J W Bosch
Department of Pathology, VU University Medical Center, Amsterdam, The Netherlands
Clin Colorectal Cancer 10:8-23. 2011..Evaluation in large well-controlled randomized trials is the next step needed to take molecular markers for CRC screening to the next level and warrant implementation in a screening setting...
Vascular endothelial growth factor-165 overexpression stimulates angiogenesis and induces cyst formation and macrophage infiltration in human ovarian cancer xenograftsMonique C A Duyndam
Department of Medical Oncology, Vrije Universiteit Medical Centre, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
Am J Pathol 160:537-48. 2002..These data provide functional evidence for a role of VEGF(165) in cyst formation and monocyte/macrophage infiltration...
Immunologic and biologic properties of the primary tumor during prolonged neoadjuvant chemoimmunotherapyEvelien Bodar
Department of Medical Oncology, VU Medical Centre, Amsterdam, The Netherlands
Oncology (Williston Park) 16:32-9. 2002..Aside from investigations concerning the immune system, other biologic processes, such as tumor angiogenesis, are being investigated at the same time...
Variation in the kinetics of caspase-3 activation, Bcl-2 phosphorylation and apoptotic morphology in unselected human ovarian cancer cell lines as a response to docetaxelGeertruida M Kolfschoten
Department of Medical Oncology, Vrije Universiteit Medical Centre, Amsterdam, The Netherlands
Biochem Pharmacol 63:733-43. 2002..We conclude that docetaxel is able to activate caspase-3, induce Bcl-2 phosphorylation and apoptosis in cells that show a prolonged G2/M arrest, but cells may also die by a caspase-3-independent cell death mechanism...
The role of VEGF in oncology: effects on hemostasis and thrombosisHerbert M Pinedo
Department of Medical Oncology, VUMC, Amsterdam, The Netherlands
Pathophysiol Haemost Thromb 33:11-2. 2003
A doxorubicin-CNGRC-peptide conjugate with prodrug propertiesYvette van Hensbergen
Department of Medical Oncology, Vrije Universiteit Medical Centre, P.O. Box 7057, 1007 MB, Amsterdam, The Netherlands
Biochem Pharmacol 63:897-908. 2002..More research is needed to identify the optimal specific chemical configuration of DOX-peptide conjugates for in vivo targeting and receptor-mediated cellular uptake...
Determinants of resistance to 2',2'-difluorodeoxycytidine (gemcitabine)Andries M Bergman
Department of Medical Oncology, VU University Medical Center, Amsterdam, The Netherlands
Drug Resist Updat 5:19-33. 2002..However, the only strong correlations with gemcitabine sensitivity are dCK activity and dFdCTP pools, with a potential important role for ribonucleotide reductase...
Efficient and selective gene transfer into primary human brain tumors by using single-chain antibody-targeted adenoviral vectors with native tropism abolishedVictor W van Beusechem
Division of Gene Therapy, Department of Medical Oncology, Vrije Universiteit Medical Center, Amsterdam, The Netherlands
J Virol 76:2753-62. 2002..Hence, single-chain targeted doubly ablated adenoviral vectors are promising tools for cancer gene therapy. They should provide an improved therapeutic index with efficient tumor transduction and effective protection of normal tissue...
Multiple mechanisms of resistance to methotrexate and novel antifolates in human CCRF-CEM leukemia cells and their implications for folate homeostasisRobert Mauritz
Department of Medical Oncology, VU Medical Center, Amsterdam, The Netherlands
Biochem Pharmacol 63:105-15. 2002....
Selective decrease in circulating V alpha 24+V beta 11+ NKT cells during HIV type 1 infectionHans J J van der Vliet
Department of Medical Oncology, Pathology, and Internal Medicine, Free University Medical Center, De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands
J Immunol 168:1490-5. 2002..In this longitudinal study no evidence was found to support an important role of Valpha24+Vbeta11+ NKT cells in determining the rate of progression during HIV-1 infection...
Design, synthesis, and biological evaluation of a dual tumor-specific motive containing integrin-targeted plasmin-cleavable doxorubicin prodrugFranciscus M H de Groot
Department of Organic Chemistry, NSR Center for Molecular Structure, Design and Synthesis, University of Nijmegen, 6525 ED Nijmegen, The Netherlands
Mol Cancer Ther 1:901-11. 2002..On the basis of these in vitro results, derivatives of 1 with improved water solubility are considered good candidates for additional development and in vivo evaluation of this dual targeting concept...
Dose-finding and pharmacokinetic study of cisplatin, gemcitabine, and SU5416 in patients with solid tumorsBart C Kuenen
Departments of Medical Oncology and Pulmonology, Vrije Universiteit Medical Center
J Clin Oncol 20:1657-67. 2002..CONCLUSION: The incidence of thromboembolic events, possibly related to the particular regimen tested in this study, discourages further investigation of this regimen...
Inhibition of angiogenesis in cancer patientsHenk M W Verheul
Dept of Internal Medicine, University Medical Center, Utrecht, The Netherlands
Expert Opin Emerg Drugs 10:403-12. 2005..In combination with chemotherapy, other serious side effects, such as bleeding and thrombosis, also occur. Here, the preclinical and clinical data of antiangiogenic agents in clinical trials at this moment are summarised...
Use of a targeted oncolytic poxvirus, JX-594, in patients with refractory primary or metastatic liver cancer: a phase I trialByeong Ho Park
Dong A University College of Medicine, Busan, South Korea
Lancet Oncol 9:533-42. 2008..We aimed to assess intratumoral injection of JX-594 in patients with refractory primary or metastatic liver cancer...
High-dose 5-Fluorouracil with uridine-diphosphoglucose rescue increases thymidylate synthase inhibition but not 5-Fluorouracil incorporation into RNA in murine tumorsGiovanni Codacci-Pisanelli
Department of Internal Medicine, University La Sapienza, Rome, Italy
Oncology 62:363-70. 2002..Since preliminary results indicate that UDPG is well tolerated by patients, the use of higher 5FU doses may improve the response rate of human tumors...
The importance of platelet counts and their contents in cancerHenk M W Verheul
Clin Cancer Res 9:3219-21. 2003
Possible molecular mechanisms involved in the toxicity of angiogenesis inhibitionHenk M W Verheul
University Medical Center Utrecht, Heidelberglaan 100, 3584 CX, Utrecht, The Netherlands
Nat Rev Cancer 7:475-85. 2007..In addition, understanding the molecular mechanisms involved in the toxicity of angiogenesis inhibition should allow more specific and more potent inhibitors to be developed...
