Research Topics
| Walter E MullerSummaryAffiliation: Frankfurt am Main Country: Germany Publications
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Detail Information
Publications
Membrane-disordering effects of beta-amyloid peptidesW E Muller
Department of Pharmacology, Biocenter University of Frankfurt, Marie Curie Strasse 9, D 60439 Frankfurt, Germany
Biochem Soc Trans 29:617-23. 2001..By contrast, membrane properties at the level of the polar heads of the phospholipid bilayer at the interface with membrane proteins are much less affected...
Neuropharmacology of the anxiolytic drug opipramol, a sigma site ligandW E Muller
Department of Pharmacology, Biocenter University Frankfurt, Marie Curie Strasse 9, D 60439 Frankfurt, Germany
Pharmacopsychiatry 37:S189-97. 2004....
Current St John's wort research from mode of action to clinical efficacyWalter E Muller
Department of Pharmacology, Biocenter JW Goethe University, Marie Curie Street 9, 60439, Frankfurt, Germany
Pharmacol Res 47:101-9. 2003..John's wort extract as an antidepressant are supported by a large number of scientific publications. Within the wide range of components in St. John's wort extract, hyperforin plays an important, if not an outstanding role...
Aging sensitizes toward ROS formation and lipid peroxidation in PS1M146L transgenic miceKatrin Schuessel
Department of Pharmacology, Biocentre, University of Frankfurt, Germany
Free Radic Biol Med 40:850-62. 2006..Hence, oxidative stress caused by the combined effects of aging and PS1 mutations may be causative for triggering neurodegenerative events in FAD patients...
Stabilization of mitochondrial function by Ginkgo biloba extract (EGb 761)Reham Abdel Kader
Department of Pharmacology, ZAFES, Biocenter, University of Frankfurt, Germany
Pharmacol Res 56:493-502. 2007..The single components of EGb 761 showed in both cell models protection of the mitochondrial membrane potential indicating that a complementary action of the components is responsible for the versatile actions of EGb 761...
Modulation of cholesterol, farnesylpyrophosphate, and geranylgeranylpyrophosphate in neuroblastoma SH-SY5Y-APP695 cells: impact on amyloid beta-protein productionGero P Hooff
Department of Pharmacology, Goethe University, Campus Riedberg, Biocenter N260, Max von Laue St 9, 60438, Frankfurt, Germany
Mol Neurobiol 41:341-50. 2010....
Mitochondrial dysfunction: the first domino in brain aging and Alzheimer's disease?Kristina Leuner
Department of Pharmacology, ZAFES, Biocenter, University of Frankfurt, Germany
Antioxid Redox Signal 9:1659-75. 2007..Herein, the authors suggest that mitochondrial protection and subsequent reduction of oxidative stress are important components of the neuroprotective activity of Ginkgo biloba extract...
Plant derived omega-3-fatty acids protect mitochondrial function in the brainGunter P Eckert
Department of Pharmacology, Campus Riedberg, Biocenter, University of Frankfurt, Germany
Pharmacol Res 61:234-41. 2010....
Hyperforin modifies neuronal membrane properties in vivoGunter P Eckert
Institute of Pharmacology, J W Goethe University, Biocenter N260, Marie Curie Strasse 9, 60439 Frankfurt, Germany
Neurosci Lett 367:139-43. 2004..Our data emphasises a membrane interaction of hyperforin that possibly contributes to its pharmacological effects...
Ginkgo biloba extract (EGb761) influences monoaminergic neurotransmission via inhibition of NE uptake, but not MAO activity after chronic treatmentChristian J Fehske
Department of Pharmacology, ZAFES, Biocenter, University of Frankfurt, Frankfurt, Germany
Pharmacol Res 60:68-73. 2009....
Increased apoptotic cell death in sporadic and genetic Alzheimer's diseaseAnne Eckert
Department of Pharmacology, Biocenter, University of Frankfurt, 60439 Frankfurt am Main, Germany
Ann N Y Acad Sci 1010:604-9. 2003..Finally, we propose a hypothetical sequence of the pathogenic steps linking sporadic AD, FAD, Abeta production, mitochondrial dysfunction with caspase pathway, and neuronal loss...
Isoprenoids, small GTPases and Alzheimer's diseaseGero P Hooff
Department of Pharmacology, Campus Riedberg, Goethe University, 60438 Frankfurt, Germany
Biochim Biophys Acta 1801:896-905. 2010....
Liposome-incorporated DHA increases neuronal survival by enhancing non-amyloidogenic APP processingGunter P Eckert
Department of Pharmacology, Goethe University, Biocenter, D 60438 Frankfurt, Germany
Biochim Biophys Acta 1808:236-43. 2011..Our data suggest that liposomal DHA is able to restore or maintain physiological membrane properties, which are required for neuroprotective sAPP? secretion and autocrine modulation of neuronal survival...
Regulation of the brain isoprenoids farnesyl- and geranylgeranylpyrophosphate is altered in male Alzheimer patientsGunter P Eckert
Department of Pharmacology, Biocenter Niederursel, University of Frankfurt, Campus Riedberg, Max von Laue St 9, Frankfurt 60438, Germany
Neurobiol Dis 35:251-7. 2009..A tentative conclusion is that if indeed regulation of FPP and GGPP is altered in AD brain such changes may stimulate protein prenylation and contribute to AD neuropathophysiology...
A rapid and sensitive assay for determining human brain levels of farnesyl-(FPP) and geranylgeranylpyrophosphate (GGPP) and transferase activities using UHPLC-MS/MSGero P Hooff
Department of Pharmacology, Biocenter Niederursel, University of Frankfurt, Max von Laue Str 9, 60438 Frankfurt, Germany
Anal Bioanal Chem 398:1801-8. 2010....
Mitochondrial dysfunction: common final pathway in brain aging and Alzheimer's disease--therapeutic aspectsWalter E Muller
Department of Pharmacology, Biocenter, University of Frankfurt, Max von Laue Strasse 9, 60438, Frankfurt, Germany
Mol Neurobiol 41:159-71. 2010..We suggest that mitochondrial protection and subsequent reduction of oxidative stress are important targets for prevention and long-term treatment of early stages of AD...
Cytoprotective effects of olive mill wastewater extract and its main constituent hydroxytyrosol in PC12 cellsSebastian Schaffer
Institute of Pharmacology, Biocenter Niederursel, University of Frankfurt, Max von Laue Strasse 9, 60438 Frankfurt am Main, Germany
Pharmacol Res 62:322-7. 2010..Furthermore, correlation analyses revealed that the observed cytoprotective effects in PC12 cells are likely due to HT present in the extract...
Mitochondrial dysfunction, apoptotic cell death, and Alzheimer's diseaseAnne Eckert
Department of Pharmacology, Biocenter, J W Goethe University of Frankfurt, Marie Curie Str 9, D 60439 Frankfurt am Main, Germany
Biochem Pharmacol 66:1627-34. 2003..Finally, we emphasize a hypothetical sequence of the pathogenic steps linking sporadic AD, FAD, and Abeta production with mitochondrial dysfunction, caspase pathway, and neuronal loss...
Isoprenoid quantitation in human brain tissue: a validated HPLC-fluorescence detection method for endogenous farnesyl- (FPP) and geranylgeranylpyrophosphate (GGPP)Gero P Hooff
Department of Pharmacology, Biocenter Niederursel, University of Frankfurt, Max von Laue Str 9, 60438, Frankfurt, Germany
Anal Bioanal Chem 392:673-80. 2008..Overall, this new method introduces the ability to simultaneously quantify FPP and GGPP in human brain tissue, and is potentially applicable to several other tissues and species...
The interaction of beta-amyloid protein with cellular membranes stimulates its own productionImke Peters
Department of Pharmacology, Goethe University of Frankfurt am Main, Campus Riedberg, Biocenter Geb N260, R 1 09, Max von Laue Str 9, D 60438 Frankfurt, Germany
Biochim Biophys Acta 1788:964-72. 2009..Based on our novel findings, we propose that oligoAbeta((1-40)) accelerates the proteolytic cleavage of APP by decreasing membrane fluidity...
Bcl-2 upregulation and neuroprotection in guinea pig brain following chronic simvastatin treatmentCornelia Franke
Department of Pharmacology, ZAFES, Biocenter Niederursel, N260 Max von Laue Str 9, University of Frankfurt, Germany
Neurobiol Dis 25:438-45. 2007..These results provide new insight into potential mechanisms for the protective actions of statins within the CNS where programmed cell death has been implicated...
Impact of aging: sporadic, and genetic risk factors on vulnerability to apoptosis in Alzheimer's diseaseKatharina Schindowski
Department of Pharmacology, Biocenter, J.W. Goethe University of Frankfurt, Marie-Curie-Str. 9, D-60439 Frankfurt am Main, Germany
Neuromolecular Med 4:161-78. 2003..In contrast, normal aging results in an increased susceptibility to apoptosis of both, CD4+ and CD8+ T cells...
Treatment duration (persistence) of basal insulin supported oral therapy (BOT) in Type-2 diabetic patients: comparison of insulin glargine with NPH insulinRenate Quinzler
DAPI German Institute for Drug Use Evaluation, Eschborn, Germany
Int J Clin Pharmacol Ther 50:24-32. 2012..To compare the persistence (treatment duration) of basal insulin supported oral therapy (BOT) using insulin glargine (GLA) or NPH insulin (NPH) in Type-2 diabetic patients...
Increased T-cell reactivity and elevated levels of CD8+ memory T-cells in Alzheimer's disease-patients and T-cell hyporeactivity in an Alzheimer's disease-mouse model: implications for immunotherapyKatharina Schindowski
Institute of Pharmacology, Biocenter building N260, Johann Wolfgang Goethe University, Max von Laue Strasse 9, 60438 Frankfurt am Main, Germany
Neuromolecular Med 9:340-54. 2007..Our data implicate the generation of reactive memory T-cell in AD and of anergic memory T-cells in transgenic mice and should be taken into concern when designing immunotherapy...
Impaired Cu/Zn-SOD activity contributes to increased oxidative damage in APP transgenic miceKatrin Schuessel
Department of Pharmacology, Biocentre, J W Goethe University of Frankfurt, Germany
Neurobiol Dis 18:89-99. 2005..Our results demonstrate that impaired Cu/Zn-SOD activity contributes to oxidative damage in Thy1-APP751(SL) transgenic mice, and these findings are closely linked to increased beta-amyloidogenic cleavage of APP...
Cholesterol: Coupling between membrane microenvironment and ABC transporter activitySascha Meyer dos Santos
Department of Pharmacology, ZAFES, Biocenter Niederursel, N260, Max von Laue Str 9, University of Frankfurt, Germany
Biochem Biophys Res Commun 354:216-21. 2007..Enrichment of membrane cholesterol changed lipid raft distribution but not the localisation of Pgp. From our data we conclude that Pgp-transport capacity depends on accurate lipid raft properties...
Cholesterol modulates amyloid beta-peptide's membrane interactionsGunter P Eckert
Department of Pharmacology, Biocenter Niederursel, University of Frankfurt, Germany
Pharmacopsychiatry 36:S136-43. 2003..Thus, elucidation of the structure and function of different cholesterol pools is necessary in understanding the coherence between cholesterol and AD...
Stabilization of mitochondrial membrane potential and improvement of neuronal energy metabolism by Ginkgo biloba extract EGb 761Anne Eckert
Department of Pharmacology, Biocenter, University of Frankfurt, Germany
Ann N Y Acad Sci 1056:474-85. 2005..Taken together, our findings clearly show stabilization and protection of mitochondrial function as a specific and very sensitive property of EGb 761 at therapeutically relevant doses...
Presenilin 1 modifies lipid raft composition of neuronal membranesGunter P Eckert
Department of Pharmacology, ZAFES, Campus Riedberg, Biocenter Niederursel, University of Frankfurt, Frankfurt, Germany
Biochem Biophys Res Commun 382:673-7. 2009..Moreover, our data reveal significant changes in membrane micro-domains and indicate that PS1 induces the formation of lipid rafts...
The amyloid precursor protein protects PC12 cells against endoplasmic reticulum stress-induced apoptosisDonat Kogel
Interdisciplinary Center for Clinical Research IZKF, Research Group Apoptosis and Cell Death, University Münster Clinics, Munster, Germany
J Neurochem 87:248-56. 2003..Our data indicate that APP plays an important physiological role in protecting neurons from the consequences of prolonged ER stress, and that APP mutations associated with familial Alzheimer's disease may impair this protective activity...
Mitochondrial dysfunction in sporadic and genetic Alzheimer's diseaseSusanne Hauptmann
Department of Pharmacology Biocentrs, University of Frankfurt, 60439 Frankfurt, Germany
Exp Gerontol 41:668-73. 2006....
Tocotrienols: constitutional effects in aging and diseaseSebastian Schaffer
Institute of Pharmacology ZAFES Member, Biocenter Niederursel, University of Frankfurt, Frankfurt am Main, Germany
J Nutr 135:151-4. 2005..This review summarizes the main antioxidant and nonantioxidant effects of tocotrienols and assesses their potential as health-maintaining compounds...
Amyloid beta-induced changes in nitric oxide production and mitochondrial activity lead to apoptosisUta Keil
Department of Pharmacology, Biocenter, University of Frankfurt, 60439 Frankfurt, Germany
J Biol Chem 279:50310-20. 2004..We suggest a hypothetical sequence of pathogenic steps linking mutant APP expression and amyloid production with enhanced NO production and mitochondrial dysfunction finally leading to cell death...
Hyperforin activates nonselective cation channels (NSCCs)Kristina Treiber
Department of Pharmacology, Biocenter, N260, University of Frankfurt, Marie-Curie-Str. 9, 60439 Frankfurt, Germany
Br J Pharmacol 145:75-83. 2005..British Journal of Pharmacology (2005) 145, 75-83. doi:10.1038/sj.bjp.0706155...
Piracetam improves mitochondrial dysfunction following oxidative stressUta Keil
Department of Pharmacology, Biocenter, N260, University of Frankfurt, Marie-Curie-Strasse 9, 60439 Frankfurt, Germany
Br J Pharmacol 147:199-208. 2006..Mitochondrial stabilization and protection might be an important mechanism to explain many of piracetam's beneficial effects in elderly patients...
Reduction of trophic support enhances apoptosis in PC12 cells expressing Alzheimer's APP mutation and sensitizes cells to staurosporine-induced cell deathSteffen Leutz
Department of Pharmacology, Biocenter, University of Frankfurt, Germany
J Mol Neurosci 18:189-201. 2002..Our study further emphasizes the pathogenic role of mutant APP and may provide new insights in the mechanisms underlying the massive neurodegeneration in brain from patients bearing the APPsw mutation...
Enhancement of proteolytic processing of the beta-amyloid precursor protein by hyperforinBettina Froestl
Department of Pharmacology, Biocenter, University of Frankfurt, Marie-Curie-Str. 9, D-60439 Frankfurt, Germany
Biochem Pharmacol 66:2177-84. 2003..These results suggest that hyperforin is an activator of secretory processing of APP with a novel mechanism of action not solely dependent on its effects on intracellular pH...
Mitochondrial dysfunction induced by disease relevant AbetaPP and tau protein mutationsUta Keil
Department of Pharmacology, Biocenter, University of Frankfurt, 60439 Frankfurt, Germany
J Alzheimers Dis 9:139-46. 2006..Thus, both Alzheimer relevant protein alterations seem to have synergistic actions probably at the level of mitochondria leading to synaptic dysfunction and apoptotic cell death...
Hydroxytyrosol-rich olive mill wastewater extract protects brain cells in vitro and ex vivoSebastian Schaffer
Institute of Pharmacology ZAFES, Biocenter Niederursel, University of Frankfurt, 60438 Frankfurt am Main, Germany
J Agric Food Chem 55:5043-9. 2007..In synthesis, the ex vivo data provide the first evidence of neuroprotective effects of oral hydroxytyrosol intake. Keywords: Hydroxytyrosol; olive mill wastewater; dissociated brain cells; oxidative stress; brain; Mediterranean diet...
Lipid rafts of purified mouse brain synaptosomes prepared with or without detergent reveal different lipid and protein domainsGunter P Eckert
Department of Pharmacology, Biocenter Niederursel, University of Frankfurt, Marie-Curie-Str. 9, D-60439, Frankfurt, Germany
Brain Res 962:144-50. 2003..Lipid rafts from the nerve terminal of neurons prepared with or without detergents may represent different membrane domains each with unique specialized functions...
Generic switch after ramipril patent expiry is not associated with decreased pharmacy refill compliance: a retrospective study using the DAPI databaseMiriam Ude
Department of Pharmacology, Goethe University Frankfurt, Frankfurt am Main, Germany
J Hypertens 29:1837-45. 2011..The purpose of this study was to evaluate whether switching from brand name ramipril to a generic product after patent expiry may negatively affect patients' refill compliance...
Age-related impairment of human T lymphocytes' activation: specific differences between CD4(+) and CD8(+) subsetsKatharina Schindowski
Department of Pharmacology, Johann Wolfgang Goethe University Biocenter, Marie Curie Strasse 9, 60439 Frankfurt Main, Germany
Mech Ageing Dev 123:375-90. 2002..The results will be discussed in relation to their relevance in neurodegenerative and psychiatric disorders...
Neurotoxic mechanisms caused by the Alzheimer's disease-linked Swedish amyloid precursor protein mutation: oxidative stress, caspases, and the JNK pathwayCelio A Marques
Department of Pharmacology, Biocenter, University of Frankfurt, 60439 Frankfurt, Germany
J Biol Chem 278:28294-302. 2003....
Reduced TRPC channel expression in psoriatic keratinocytes is associated with impaired differentiation and enhanced proliferationKristina Leuner
Institute of Pharmacology, Biocenter Niederursel, Johann Wolfgang Goethe University, Frankfurt, Germany
PLoS ONE 6:e14716. 2011..As TRPC6 channel activation can partially overcome this Ca(2+) entry defect, specific TRPC channel activators may be potential new drug candidates for the topical treatment of psoriasis...
Effects of antidepressants on the brain/plasma distribution of corticosteroneClaudia-Carolin Weber
Department of Pharmacology, Biocenter (ZAFES, University of Frankfurt, Frankfurt, Germany
Neuropsychopharmacology 31:2443-8. 2006..In addition, St John's wort is the only antidepressant tested which slightly elevated Pgp protein level in the brain...
[Tricyclics as co-analgesics. Therapeutic options for chronic pain]Kristina Leuner
, Biozentrum Niederursel, Max-von-Laue-Str. 9, 60438 Frankfurt am Main
Pharm Unserer Zeit 37:220-5. 2008
