Research Topics
| Jian Xin LiSummaryAffiliation: Nanjing University Country: China Publications
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Detail Information
Publications
Five new oleanolic acid glycosides from Achyranthes bidentata with inhibitory activity on osteoclast formationJian Xin Li
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, P R China
Planta Med 71:673-9. 2005..All the oleanolic acid glycosides inhibited the formation of osteoclast-like multinucleated cells (OCLs) induced by 1alpha,25(OH)2D3 in a co-culture assay system...
Cimicifugae rhizoma: from origins, bioactive constituents to clinical outcomesJian Xin Li
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, 22 Hankou Road, Nanjing, 210093, China
Curr Med Chem 13:2927-51. 2006....
Triterpenoids from Cimicifugae rhizoma, a novel class of inhibitors on bone resorption and ovariectomy-induced bone lossJ X Li
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, PR China
Maturitas 58:59-69. 2007....
An unusual metabolite of cimicidol-3-O-beta-D-xyloside from Cimicifugae rhizoma by rat intestinal bacteriaJian Xin Li
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, PR China
Chem Biodivers 5:290-8. 2008....
Osteoprotective effect of extract from Achyranthes bidentata in ovariectomized ratsCui Cui He
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, China
J Ethnopharmacol 127:229-34. 2010..The present study is to clarify the fractions responsible for the activity and further explore the osteoprotective effect of the fraction in vivo...
Synthesis and biological evaluation of unique stereodimers of sinomenine analogues as potential inhibitors of NO productionPeng Teng
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, PR China
Bioorg Med Chem 19:3096-104. 2011..Interestingly, (S)-dimers displayed a better bioactivity than (R)-dimers. These compounds may sever as lead candidates in the development of novel therapeutic drugs for RA treatment...
Glycoside modification of oleanolic acid derivatives as a novel class of anti-osteoclast formation agentsJun Feng Li
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, PR China
Carbohydr Res 344:599-605. 2009..The structure-activity relationships of these compounds were also discussed...
Synthesis and biological evaluation of novel sinomenine derivatives as anti-inflammatory agentsPeng Teng
State Key Laboratory of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, 210093, PR China
Eur J Med Chem 50:63-74. 2012..Moreover, 3b and 2f significantly alleviated the lipopolysaccharide (LPS)-induced mortality. These two compounds might serve as valuable candidates for anti-inflammatory drug discovery...
Biocatalyzed cross-coupling of sinomenine and guaiacol by Antrodiella semisupinaZhang Shuang Deng
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, 210093, P R China
Org Lett 10:1119-22. 2008..4 exhibited more potent inhibitory activity on IL-6 production than 1 in human synovial sarcoma cell (SW982), and 5 stimulated IL-6 production...
Quinoxaline derivative of oleanolic acid inhibits osteoclastic bone resorption and prevents ovariectomy-induced bone lossYu Zhao
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, China
Menopause 18:690-7. 2011..The aim of the present study was to evaluate the activities of QOA-8a on bone resorption in vitro and its osteoprotective effect in vivo...
Synthesis of a novel series of diphenolic chromone derivatives as inhibitors of NO production in LPS-activated RAW264.7 macrophagesGuo Biao Liu
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, China
Bioorg Med Chem 18:2864-71. 2010..Furthermore, a computational analysis of physicochemical parameters revealed that the most of the compounds possessed drug-like properties...
A novel synthetic oleanolic acid derivative with amino acid conjugate suppresses tumour growth by inducing cell cycle arrestXiao Min Lu
State Key Laboratory of Pharmaceutical Biotechnology, School of Life Sciences, Nanjing University, 22 Hankou Road, Nanjing, 210093, China
J Pharm Pharmacol 59:1087-93. 2007..OA did not show such activities. These results suggest that AOA-GMe may induce growth arrest in tumour cells through regulation of proteins involved in the cell cycle...
Synthesis and evaluation of a novel series of heterocyclic oleanolic acid derivatives with anti-osteoclast formation activityJun Feng Li
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, China
Eur J Med Chem 44:2796-806. 2009..Among the derivatives, compounds 2a and 8a displayed quite a potent activity even at 200 nM. The structure-activity relationships of the derivatives were also discussed...
pH-dependent, stereoselective dimerization of sinomenineZhang Shuang Deng
Key Laboratory of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, 210093, PR China
Org Lett 10:3879-82. 2008..The bioassay results using human synovial sarcoma cells (SW982) showed that 2 inhibited, while 3 stimulated, IL-6 production...
Synthesis and evaluation of a novel series of quinoline derivatives with immunosuppressive activityGuo Biao Liu
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, China
Bioorg Med Chem 17:5433-41. 2009....
Inhibitory effects of citrus extracts on the experimental pulmonary fibrosisXian Mei Zhou
Department of Respiratory Medicine, Affiliated Jiangsu Province Hospital of Traditional Chinese Medicine, Nanjing University of Traditional Chinese Medicine, Nanjing, China
J Ethnopharmacol 126:143-8. 2009..The present study was designed to clarify the active principles responsible for the activity and further explore the anti-pulmonary fibrosis effect in vivo...
[Isolation and identification of triterpenoids from root of Achyranthes bidentata in Henan]Shu-ping Jia
School of Chemistry and Chemical Engineering, Nanjing University, China
Zhongguo Zhong Yao Za Zhi 31:1244-7. 2006..CONCLUSION: Compounds 1 and 2 were isolated from the natural resources for the first time...
Ultrasound-promoted intramolecular direct arylation in a capillary flow microreactorLei Zhang
State Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing 210093, PR China
Ultrason Sonochem 19:250-6. 2012..The ultrasonic irritation not only greatly promoted the conversion and selectivity of the direct arylation, but also solved the clogging problem of the microreactor for solid-forming reaction and made the reaction run smoothly...
NMR-based metabonomic approach on the toxicological effects of a Cimicifuga triterpenoidCui Cui He
Key Laboratory of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University, Nanjing, 210093, People s Republic of China
J Appl Toxicol 32:88-97. 2012..The present study provides a reasonable explanation for the clinical hepatotoxicity of Cimicifuga extract...
Synthesis and activity of oleanolic acid derivatives, a novel class of inhibitors of osteoclast formationYuan Zhang
Key Lab of Analytical Chemistry for Life Science, School of Chemistry and Chemical Engineering, Nanjing University 210093, PR China
Bioorg Med Chem Lett 15:1629-32. 2005..Derivatives with proline or phenylalanine showed a tendency to enhance the inhibitory activity...
Structural revision of two flavanonol glycosides from Smilax glabraXiang Zhou
State Key Laboratory of Pharmaceutical Biotechnology, School of Life Sciences, Nanjing University, Nanjing 210093, PR China
Planta Med 75:654-5. 2009..The revised structures were determined based on intensive studies of chemical interconversion, NMR spectroscopy, and X-ray crystallographic analysis. The latest NMR data were also summarized...
Transplantation of autologous bone marrow mononuclear cells for patients with lower limb ischemiaYong quan Gu
Department of Vascular Surgery, Xuanwu Hospital, Institute of Vascular Surgery, Capital Medical University, Beijing, China
Chin Med J (Engl) 121:963-7. 2008....
